SCHEMBL5660992

SCHEMBL5660992

Cc1ccc(O)c(C2(c3cc(C)c(O)c(C)c3)C(=O)N(c3cccc(OC(F)(F)F)c3)c3ccccc32)c1

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
OPRL1 P41146 1/20 0.35
PKM P14618 1/20 0.32
CNR1 P21554 1/20 0.32
GPR55 Q9Y2T6 1/20 0.32
CETP P11597 8/20 0.32
CHRM5 P08912 2/20 0.32
EDNRB P24530 1/20 0.32
EDNRA P25101 1/20 0.32
CCKBR P32239 1/20 0.32
ADAMTS5 Q9UNA0 2/20 0.32
ADAMTS4 O75173 1/20 0.32
AMPD2 Q01433 1/20 0.31
PIM1 P11309 2/20 0.31
PIM2 Q9P1W9 2/20 0.31
TOP2A P11388 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5659652 0.91 CETP (0.34) OPRL1CETPEDNRBEDNRACCKBR
SCHEMBL5661607 0.89 OPRL1 (0.33) OPRL1CETPEDNRBEDNRACCKBR
SCHEMBL5661171 0.89 ADAMTS5 (0.39) PKMCNR1GPR55ADAMTS5ADAMTS4
SCHEMBL5659320 0.88 CNR1 (0.37) PKMCNR1GPR55ADAMTS5
SCHEMBL5659844 0.86 OPRL1 (0.33) OPRL1CETPEDNRBEDNRACCKBR
SCHEMBL5656691 0.82 SCN9A (0.37) OPRL1CETPCHRM5EDNRBEDNRA
SCHEMBL5661921 0.81 MAPT (0.41)
SCHEMBL5661875 0.80 SLC6A2 (0.37) PKMCNR1GPR55ADAMTS5
SCHEMBL5658260 0.79 ALDH1A1 (0.40) ADAMTS5ADAMTS4
SCHEMBL5662233 0.79 HSP90AA1 (0.41) PKMCNR1GPR55

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7250442-B2 Dihydroindol-2-one derivatives as steroid hormone nuclear receptor modulators ELI LILLY AND COMPANY (US) 2007-07-31 US disclosed
US-7250442-B2 Dihydroindol-2-one derivatives as steroid hormone nuclear receptor modulators ELI LILLY AND COMPANY (US) 2007-07-31 US disclosed
US-7250442-B2 Dihydroindol-2-one derivatives as steroid hormone nuclear receptor modulators ELI LILLY AND COMPANY (US) 2007-07-31 US disclosed
US-20050054712-A1 Dihydroindol-2-one derivatives as steroid hormone nuclear receptor modulators ELI LILLY AND COMPANY 2005-03-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050054712-A1 Dihydroindol-2-one derivatives as steroid hormone nuclear receptor modulators NR3C2, NR5A1, NR5A2 OPRL1 267/4885PKM 1991/4885CNR1 362/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.