SCHEMBL5669074

SCHEMBL5669074

CCOC(=O)C(C)(C)Oc1cc(CC[AsH2])cc(OC)c1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 4/20 0.50
PPARG P37231 2/20 0.50
CYP3A4 P08684 2/20 0.48
ABCB11 O95342 1/20 0.48
CYP1A2 P05177 1/20 0.48
TSHR P16473 1/20 0.48
HTR2A P28223 1/20 0.48
PMP22 Q01453 1/20 0.48
FBP1 P09467 8/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
PTGS2 P35354 1/20 0.38
ALDH1A1 P00352 1/20 0.36
HPGD P15428 1/20 0.36
CALM1 P0DP23 2/20 0.35
AKR1B1 P15121 1/20 0.35
MGLL Q99685 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1549802 0.87 PPARA (0.50) PPARAPPARGCYP3A4ABCB11CYP1A2
SCHEMBL1550074 0.80 PPARA (0.51) PPARAPPARGCYP3A4ABCB11CYP1A2
SCHEMBL2964422 0.78 PPARA (0.50) PPARAPPARGCYP3A4ABCB11CYP1A2
SCHEMBL12670824 0.76 PPARA (0.62) PPARAPPARGCYP3A4ABCB11CYP1A2
SCHEMBL7979408 0.75 PPARA (0.73) PPARAPPARGCYP3A4ABCB11CYP1A2
SCHEMBL1549732 0.72 FBP1 (0.72) PPARACYP3A4ABCB11CYP1A2TSHR
SCHEMBL1549729 0.72 FBP1 (0.72) PPARACYP3A4ABCB11CYP1A2TSHR
SCHEMBL3484056 0.69 PPARA (0.75) PPARAPPARGCYP3A4ABCB11CYP1A2
SCHEMBL63490 0.69 CYP4F2 (0.56) CYP3A4TSHRSMN1; SMN2ALDH1A1HPGD
SCHEMBL6093013 0.69 PPARA (0.70) PPARAPPARGCYP3A4ABCB11CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1682508-A1 PHENYL DERIVATIVES AS PPAR AGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2006-07-26 EP disclosed
WO-2005049573-A1 PHENYL DERIVATIVES AS PPAR AGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2005-06-02 WO disclosed