SCHEMBL5669352

SCHEMBL5669352

OC(CNC(c1cccc(Oc2ccc(F)cc2)c1)c1cccc(C(F)(F)C(F)(F)F)c1)C(F)(F)F

nearest known ligand 0.40

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CETP P11597 12/20 0.40
SLC6A9 P48067 1/20 0.34
SCN8A Q9UQD0 1/20 0.34
SCN10A Q9Y5Y9 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5669140 1.00 CETP (0.40) CETPSLC6A9SCN8ASCN10A
SCHEMBL6277527 0.94 CETP (0.39) CETPSLC6A9
SCHEMBL1903178 0.94 CETP (0.39) CETPSLC6A9
SCHEMBL992083 0.93 CETP (0.43) CETP
SCHEMBL6280371 0.93 CETP (0.43) CETP
SCHEMBL5670346 0.92 CETP (0.41) CETP
SCHEMBL6568915 0.92 CETP (0.41) CETP
SCHEMBL5670800 0.91 CETP (0.44) CETP
SCHEMBL6568898 0.91 CETP (0.44) CETP
SCHEMBL5668806 0.89 CETP (0.41) CETP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1670446-A2 METHOD OF INHIBITING REMNANT LIPOPROTEIN PRODUCTION JAPAN TOBACCO INC. (JP) 2006-06-21 EP claimed
WO-2005030185-A2 METHOD OF INHIBITING REMNANT LIPOPROTEIN PRODUCTION JAPAN TOBACCO INC. (JP) 2005-04-07 WO claimed
WO-2005117869-A1 COMBINATIONS COMPRISING (S)-AMLODIPINE AND A CHOLESTERYL ESTER TRANSFER PROTEIN INHIBITOR, AND METHODS FOR REDUCING HYPERTENSION SEPRACOR INC. (US) 2005-12-15 WO disclosed
EP-1401399-A2 PHARMACEUTICAL COMPOSITIONS CONTAINING POLYMER AND DRUG ASSEMBLIES Pfizer Products Inc. (US) 2004-03-31 EP disclosed
WO-2003000226-A2 PHARMACEUTICAL COMPOSITIONS CONTAINING POLYMER AND DRUG ASSEMBLIES PFIZER PRODUCTS INC. (US) 2003-01-03 WO disclosed