SCHEMBL5683223

SCHEMBL5683223

COc1cc(-c2nccc(CCl)n2)cc(OC)c1OC

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.42
TSHR P16473 2/20 0.42
CYP1A1 P04798 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2E1 P05181 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C8 P10632 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2A6 P11509 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP4B1 P13584 1/20 0.42
CYP2B6 P20813 1/20 0.42
CYP3A5 P20815 1/20 0.42
CYP2A7 P20853 1/20 0.42
CYP3A7 P24462 1/20 0.42
CYP2F1 P24903 1/20 0.42
CYP2C18 P33260 1/20 0.42
CYP2C19 P33261 1/20 0.42
CYP2J2 P51589 1/20 0.42
CYP4F2 P78329 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5679867 0.85 FYN (0.44) MAPTTSHRCYP1A1CYP1A2CYP2E1
SCHEMBL5681214 0.81 TP53 (0.52) ALDH1A1MEN1KMT2ABRD4KDM4E
SCHEMBL30263762 0.80 TSHR (0.47) MAPTTSHRCYP1A1CYP1A2CYP2E1
SCHEMBL28985313 0.80 TSHR (0.47) MAPTTSHRCYP1A1CYP1A2CYP2E1
SCHEMBL5679879 0.79 SYK (0.47) SYKALDH1A1BRD4KDM4ETDP1
SCHEMBL30263736 0.78 CYP1A1 (0.46) MAPTTSHRCYP1A1CYP1A2CYP2E1
SCHEMBL5679981 0.78 CYP1A1 (0.46) MAPTTSHRCYP1A1CYP1A2CYP2E1
SCHEMBL28985316 0.78 CYP1A1 (0.46) MAPTTSHRCYP1A1CYP1A2CYP2E1
SCHEMBL5682153 0.78 TP53 (0.49) TSHRCYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL5679729 0.75 BRD4 (0.47) MAPTTSHRALDH1A1NPC1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1403249-B1 CYCLIC DIAMINE COMPOUNDS BEARING SIX-MEMBERED CYCLIC GROUPS KOWA CO (JP) 2006-03-15 EP disclosed
EP-1403249-A1 CYCLIC DIAMINE COMPOUNDS BEARING SIX-MEMBERED CYCLIC GROUPS Kowa Co., Ltd. (JP) 2004-03-31 EP disclosed
US-6509329-B1 Inhibitory effects on both cell adhesion and cell infiltration and is useful as a medicine for prevention or treatment of diseases such as allergy, asthma, rheumatism, arteriosclerosis and inflammation KOWA CO., LTD. (JP) 2003-01-21 US disclosed