SCHEMBL5684178

SCHEMBL5684178

CCCCc1ccc2c(c1)CCc1cc(-c3ccc(C#N)cc3)ccc1-2

nearest known ligand 0.57

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.57
HSD17B10 Q99714 1/20 0.57
HRH3 Q9Y5N1 12/20 0.49
MPL P40238 4/20 0.41
KCNH2 Q12809 1/20 0.40
CYP2A6 P11509 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5686555 0.96 TSHR (0.63) TSHRHSD17B10HRH3MPLKCNH2
SCHEMBL5683341 0.95 TSHR (0.66) TSHRHSD17B10HRH3
SCHEMBL5683932 0.95 TSHR (0.66) TSHRHSD17B10HRH3
SCHEMBL5884950 0.92 TSHR (0.57) TSHRHSD17B10HRH3MPLKCNH2
SCHEMBL5683927 0.92 HRH3 (0.51) TSHRHSD17B10HRH3KCNH2CYP2A6
SCHEMBL5684587 0.88 TSHR (0.63) TSHRHSD17B10HRH3CYP2A6
SCHEMBL5683706 0.87 TSHR (0.66) TSHRHSD17B10HRH3
SCHEMBL5686753 0.87 TSHR (0.66) TSHRHSD17B10HRH3
SCHEMBL5687633 0.86 CYP2A6 (0.51) TSHRHSD17B10HRH3KCNH2CYP2A6
SCHEMBL5683748 0.84 HRH3 (0.51) TSHRHSD17B10HRH3KCNH2CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100422124-C Fused ring compound DAINIPPON INK & CHEMICALS (JP) 2008-10-01 CN disclosed
US-7067179-B1 Fused ring compound DAINIPPON INK AND CHEMICALS, INC. (JP) 2006-06-27 US disclosed
EP-1201632-B1 FUSED RING COMPOUND DAINIPPON INK & CHEMICALS (JP) 2006-03-29 EP disclosed
EP-1201632-A1 FUSED RING COMPOUND DAINIPPON INK AND CHEMICALS, INC. (JP) 2002-05-02 EP disclosed