SCHEMBL5684335

SCHEMBL5684335

CCCc1ccc2c(ccc3cc(-c4ccc(OC(F)(F)F)cc4)ccc32)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 1/20 0.42
CHRNA7 P36544 1/20 0.39
HRH3 Q9Y5N1 4/20 0.39
TSHR P16473 1/20 0.39
NCEH1 Q6PIU2 2/20 0.38
JAK2 O60674 1/20 0.38
ROCK2 O75116 1/20 0.38
PRKD3 O94806 1/20 0.38
PRKCG P05129 1/20 0.38
PHKG2 P15735 1/20 0.38
RPS6KB1 P23443 1/20 0.38
MARK3 P27448 1/20 0.38
PRKCI P41743 1/20 0.38
CLK2 P49760 1/20 0.38
IRAK1 P51617 1/20 0.38
RPS6KA3 P51812 1/20 0.38
PRKCD Q05655 1/20 0.38
MAP4K2 Q12851 1/20 0.38
STK3 Q13188 1/20 0.38
CAMK2B Q13554 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3158489 0.94 TSHR (0.42) GSK3BCHRNA7HRH3TSHRJAK2
SCHEMBL3158383 0.94 TSHR (0.42) GSK3BCHRNA7HRH3TSHRJAK2
SCHEMBL7664905 0.89 NCEH1 (0.40) TSHRNCEH1KIF11
SCHEMBL3170923 0.86 GSK3B (0.37) GSK3BCHRNA7TSHRNCEH1SERPINE1
SCHEMBL3168983 0.86 PCSK9 (0.43) GSK3BCHRNA7HRH3TSHRJAK2
SCHEMBL3166994 0.86 PCSK9 (0.43) GSK3BCHRNA7HRH3TSHRJAK2
SCHEMBL3165349 0.86 SLC13A5 (0.43) GSK3BCHRNA7TSHRJAK2ROCK2
SCHEMBL3162115 0.86 SLC13A5 (0.43) GSK3BCHRNA7TSHRJAK2ROCK2
SCHEMBL6059636 0.85 GSK3B (0.39) GSK3BCHRNA7TSHRSERPINE1GRM2
SCHEMBL5684909 0.85 GRM2 (0.36) GSK3BCHRNA7TSHRNCEH1GRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7067179-B1 Fused ring compound DAINIPPON INK AND CHEMICALS, INC. (JP) 2006-06-27 US disclosed
EP-1201632-B1 FUSED RING COMPOUND DAINIPPON INK & CHEMICALS (JP) 2006-03-29 EP disclosed
EP-1201632-A1 FUSED RING COMPOUND DAINIPPON INK AND CHEMICALS, INC. (JP) 2002-05-02 EP disclosed