SCHEMBL5684693

SCHEMBL5684693

CCCC1CCc2c(ccc3c2CCC(c2ccc(C#N)c(F)c2)C3)C1

nearest known ligand 0.34

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.34
CYP2C8 P10632 1/20 0.34
S1PR3 Q99500 1/20 0.34
KDM4E B2RXH2 1/20 0.33
HTR1D P28221 2/20 0.32
HTR1B P28222 2/20 0.32
SGPL1 O95470 2/20 0.32
S1PR1 P21453 6/20 0.32
ALDH1A1 P00352 1/20 0.31
TRPV4 Q9HBA0 1/20 0.31
CHEK1 O14757 1/20 0.31
POLB P06746 1/20 0.31
DRD2 P14416 2/20 0.31
DRD3 P35462 2/20 0.31
S1PR4 O95977 1/20 0.31
S1PR5 Q9H228 1/20 0.31
FYN P06241 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5684309 0.94 CYP3A4 (0.39) CYP3A4CYP2C8S1PR3HTR1DHTR1B
SCHEMBL5683721 0.93 CYP3A4 (0.43) CYP3A4CYP2C8S1PR3SGPL1S1PR1
SCHEMBL5687011 0.92 CYP3A4 (0.44) CYP3A4CYP2C8S1PR3SGPL1S1PR1
SCHEMBL5684697 0.92 CYP3A4 (0.44) CYP3A4CYP2C8S1PR3SGPL1S1PR1
SCHEMBL5686434 0.91 TRPV4 (0.33) HTR1DHTR1BTRPV4CHEK1DRD2
SCHEMBL14526396 0.87 TRPV4 (0.33) KDM4EHTR1DHTR1BALDH1A1TRPV4
SCHEMBL5687262 0.87 HTR1D (0.38) CYP3A4CYP2C8S1PR3HTR1DHTR1B
SCHEMBL5685300 0.84 HTR1D (0.32) CYP3A4CYP2C8S1PR3KDM4EHTR1D
SCHEMBL5684282 0.84 CYP3A4 (0.35) CYP3A4CYP2C8S1PR3HTR1DHTR1B
SCHEMBL5684871 0.83 HTR1D (0.36) CYP3A4CYP2C8S1PR3HTR1DHTR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7067179-B1 Fused ring compound DAINIPPON INK AND CHEMICALS, INC. (JP) 2006-06-27 US disclosed
EP-1201632-B1 FUSED RING COMPOUND DAINIPPON INK & CHEMICALS (JP) 2006-03-29 EP disclosed
EP-1201632-A1 FUSED RING COMPOUND DAINIPPON INK AND CHEMICALS, INC. (JP) 2002-05-02 EP disclosed