SCHEMBL5685170

SCHEMBL5685170

CCCCCCCc1ccc2c(c1)Cc1cc(-c3cc(F)c(C#N)c(F)c3)c(F)cc1-2

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
RARB P10826 4/20 0.40
TSHR P16473 1/20 0.40
HSD17B10 Q99714 1/20 0.40
HTR2A P28223 3/20 0.38
DRD2 P14416 1/20 0.38
SLC6A2 P23975 1/20 0.38
HTR2C P28335 1/20 0.38
SLC6A4 P31645 1/20 0.38
RARA P10276 1/20 0.37
RARG P13631 1/20 0.37
GPR3 P46089 1/20 0.34
S1PR1 P21453 2/20 0.34
SPHK2 Q9NRA0 1/20 0.33
THRA P10827 1/20 0.33
THRB P10828 1/20 0.33
MOGAT2 Q3SYC2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5684048 1.00 RARB (0.40) RARBTSHRHSD17B10HTR2ADRD2
SCHEMBL5684136 0.99 RARB (0.38) RARBTSHRHSD17B10HTR2ADRD2
SCHEMBL5683868 0.96 RARB (0.34) RARBTSHRHSD17B10HTR2ADRD2
SCHEMBL5684151 0.91 MEN1 (0.33)
SCHEMBL5684293 0.89 TSHR (0.44) RARBTSHRHSD17B10HTR2ADRD2
SCHEMBL5684164 0.89 TSHR (0.44) RARBTSHRHSD17B10HTR2ADRD2
SCHEMBL5684072 0.88 TSHR (0.42) RARBTSHRHSD17B10HTR2ADRD2
SCHEMBL5686526 0.87 KCNJ1 (0.41) RARBTSHRHSD17B10RARARARG
SCHEMBL5684732 0.87 KCNJ1 (0.41) RARBTSHRHSD17B10RARARARG
SCHEMBL5684203 0.87 TSHR (0.54) RARBTSHRHSD17B10HTR2ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7067179-B1 Fused ring compound DAINIPPON INK AND CHEMICALS, INC. (JP) 2006-06-27 US disclosed
EP-1201632-B1 FUSED RING COMPOUND DAINIPPON INK & CHEMICALS (JP) 2006-03-29 EP disclosed
EP-1201632-A1 FUSED RING COMPOUND DAINIPPON INK AND CHEMICALS, INC. (JP) 2002-05-02 EP disclosed