SCHEMBL5685545

SCHEMBL5685545

CCCCOC(=O)n1c(-c2ccc(O)cc2)nc2c1c(=O)n(CCC)c(=O)n2CCC

nearest known ligand 0.54

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 9/20 0.54
ADORA2B P29275 11/20 0.53
GAA P10253 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1946588 0.84 ADORA2B (0.53) ADORA2AADORA2B
SCHEMBL14099409 0.77 ADORA2B (0.54) ADORA2AADORA2BL3MBTL1
SCHEMBL1946574 0.77 ADORA2B (0.45) ADORA2AADORA2B
SCHEMBL1945740 0.75 MAOB (0.44) ADORA2AADORA2B
SCHEMBL1066272 0.74 ADORA2B (0.52) ADORA2AADORA2B
SCHEMBL29402274 0.74 ADORA2B (0.60) ADORA2AADORA2B
SCHEMBL21343065 0.74 ADORA2B (0.60) ADORA2AADORA2B
SCHEMBL1946977 0.72 ADORA2B (0.67) ADORA2AADORA2B
SCHEMBL1945205 0.71 ADORA2B (0.59) ADORA2AADORA2B
SCHEMBL1944406 0.71 ADORA2B (0.51) ADORA2AADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1622908-A1 XANTHINE DERIVATIVES AS A2B ADENOSINE RECEPTOR ANTAGONISTS CV THERAPEUTICS, INC. (US) 2006-02-08 EP disclosed
WO-2004106337-A1 XANTHINE DERIVATIVES AS A2B ADENOSINE RECEPTOR ANTAGONISTS CV THERAPEUTICS, INC. (US) 2004-12-09 WO disclosed
EP-1444233-A2 A 2B? ADENOSINE RECEPTOR ANTAGONISTS CV THERAPEUTICS, INC. (US) 2004-08-11 EP disclosed
WO-2003042214-A2 A2B ADENOSINE RECEPTOR ANTAGONISTS CV THERAPEUTICS, INC. (US) 2003-05-22 WO disclosed