SCHEMBL5686705

SCHEMBL5686705

C[C@@]1(C(=O)NC(Cc2ccc([Sn](C)(C)C)cc2)C(=O)O)CCCN1S(=O)(=O)c1cc(Cl)cc(Cl)c1

nearest known ligand 0.68

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 20/20 0.68
ITGB1 P05556 13/20 0.68
ITGB7 P26010 6/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6375049 0.91 ITGA4 (0.77) ITGA4ITGB1ITGB7
SCHEMBL6367713 0.90 ITGA4 (0.71) ITGA4ITGB1ITGB7
SCHEMBL6373491 0.89 ITGA4 (0.70) ITGA4ITGB1ITGB7
SCHEMBL6296771 0.89 ITGA4 (0.70) ITGA4ITGB1ITGB7
SCHEMBL6372333 0.89 ITGA4 (0.70) ITGA4ITGB1ITGB7
SCHEMBL6368938 0.88 ITGA4 (0.68) ITGA4ITGB1ITGB7
SCHEMBL6367870 0.87 ITGA4 (0.67) ITGA4ITGB1ITGB7
SCHEMBL5686886 0.87 ITGA4 (0.67) ITGA4ITGB1ITGB7
SCHEMBL6368662 0.86 ITGA4 (0.66) ITGA4ITGB1ITGB7
SCHEMBL6375051 0.85 ITGA4 (0.85) ITGA4ITGB1ITGB7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1017382-B1 BIARYLALKANOIC ACIDS AS CELL ADHESION INHIBITORS MERCK & CO INC (US) 2006-03-01 EP disclosed
EP-1001764-A4 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO INC (US) 2005-08-24 EP disclosed
US-6903075-B1 Heterocyclic amide compounds as cell adhesion inhibitors MERCK & CO., INC. (US) 2005-06-07 US disclosed
US-6291511-B1 Biarylalkanoic acids as cell adhesion inhibitors MERCK & CO., INC. 2001-09-18 US disclosed
EP-1001764-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS Merck & Co., Inc. (a New Jersey corp.) (US) 2000-05-24 EP disclosed
WO-1999064395-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO., INC. (US) 1999-12-16 WO disclosed
WO-1998053814-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO., INC. (US) 1998-12-03 WO disclosed