SCHEMBL5686709

SCHEMBL5686709

O=C(O)[C@H](Cc1ccc(I)cc1)NC(=O)[C@@H]1CCCN1S(=O)(=O)c1cccc(F)c1

nearest known ligand 0.61

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 15/20 0.61
ITGA5 P08648 5/20 0.61
ITGA4 P13612 8/20 0.58
ITGAV P06756 6/20 0.56
ITGB7 P26010 3/20 0.55
ITGA2 P17301 1/20 0.49
ITGB3 P05106 1/20 0.45
KCNQ1 P51787 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6368195 0.94 ITGB1 (0.64) ITGB1ITGA5ITGA4ITGAVITGB7
SCHEMBL6367317 0.93 ITGB1 (0.65) ITGB1ITGA5ITGA4ITGAVITGB7
SCHEMBL6368406 0.90 ITGB1 (0.55) ITGB1ITGA5ITGA4ITGAVITGB7
SCHEMBL5686669 0.89 ITGB1 (0.58) ITGB1ITGA5ITGA4ITGAVITGB7
SCHEMBL630691 0.86 KCNQ1 (0.60) ITGB1ITGA5ITGA4ITGAVITGB7
SCHEMBL630690 0.86 KCNQ1 (0.60) ITGB1ITGA5ITGA4ITGAVITGB7
SCHEMBL5171521 0.86 KCNQ1 (0.60) ITGB1ITGA5ITGA4ITGAVITGB7
SCHEMBL5689683 0.86 ITGB1 (0.55) ITGB1ITGA5ITGA4ITGAVITGB7
SCHEMBL4957436 0.86 ITGB1 (0.58) ITGB1ITGA5ITGA4ITGAVITGB7
SCHEMBL6368166 0.86 ITGB1 (0.72) ITGB1ITGA5ITGA4ITGAVITGB7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1001764-A4 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO INC (US) 2005-08-24 EP claimed
US-6903075-B1 Heterocyclic amide compounds as cell adhesion inhibitors MERCK & CO., INC. (US) 2005-06-07 US claimed
JP-2002512625-A 2002-04-23 JP claimed
EP-1001764-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS Merck & Co., Inc. (a New Jersey corp.) (US) 2000-05-24 EP claimed
WO-1999064395-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO., INC. (US) 1999-12-16 WO claimed
WO-1998053814-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO., INC. (US) 1998-12-03 WO claimed
EP-1017382-B1 BIARYLALKANOIC ACIDS AS CELL ADHESION INHIBITORS MERCK & CO INC (US) 2006-03-01 EP disclosed
EP-1001764-A4 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO INC (US) 2005-08-24 EP disclosed
US-6903075-B1 Heterocyclic amide compounds as cell adhesion inhibitors MERCK & CO., INC. (US) 2005-06-07 US disclosed
US-6291511-B1 Biarylalkanoic acids as cell adhesion inhibitors MERCK & CO., INC. 2001-09-18 US disclosed
EP-1017382-A4 BIARYLALKANOIC ACIDS AS CELL ADHESION INHIBITORS MERCK & CO INC (US) 2000-08-30 EP disclosed
EP-1017382-A1 BIARYLALKANOIC ACIDS AS CELL ADHESION INHIBITORS Merck & Co., Inc. (a New Jersey corp.) (US) 2000-07-12 EP disclosed
EP-1001764-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS Merck & Co., Inc. (a New Jersey corp.) (US) 2000-05-24 EP disclosed
WO-1999064395-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO., INC. (US) 1999-12-16 WO disclosed
WO-1998053814-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO., INC. (US) 1998-12-03 WO disclosed
WO-1998053817-A1 BIARYLALKANOIC ACIDS AS CELL ADHESION INHIBITORS MERCK & CO., INC. (US) 1998-12-03 WO disclosed