SCHEMBL6368166

SCHEMBL6368166

O=C(O)[C@H](Cc1ccc(F)cc1)NC(=O)[C@@H]1CCCN1S(=O)(=O)c1cccc(Cl)c1

nearest known ligand 0.72

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 15/20 0.72
ITGA4 P13612 9/20 0.72
ITGB7 P26010 5/20 0.64
ITGA5 P08648 4/20 0.61
ITGAV P06756 5/20 0.54
HCRTR1 O43613 1/20 0.51
HCRTR2 O43614 1/20 0.51
MAPT P10636 1/20 0.49
THRB P10828 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
ITGA2 P17301 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6368888 0.93 ITGB1 (0.73) ITGB1ITGA4ITGB7ITGA5ITGAV
SCHEMBL6368398 0.92 ITGA4 (0.69) ITGB1ITGA4ITGB7ITGA5ITGAV
SCHEMBL6368195 0.92 ITGB1 (0.64) ITGB1ITGA4ITGB7ITGA5ITGAV
SCHEMBL5687080 0.89 ITGA4 (0.66) ITGB1ITGA4ITGB7ITGA5ITGAV
SCHEMBL6372387 0.89 ITGA4 (0.66) ITGB1ITGA4ITGB7ITGA5ITGAV
SCHEMBL6367132 0.88 ITGA4 (0.66) ITGB1ITGA4ITGB7ITGA5ITGAV
SCHEMBL6367902 0.88 ITGB1 (0.59) ITGB1ITGA4ITGB7ITGA5ITGAV
SCHEMBL6374288 0.88 ITGB1 (0.68) ITGB1ITGA4ITGB7ITGA5ITGAV
SCHEMBL6367317 0.87 ITGB1 (0.65) ITGB1ITGA4ITGB7ITGA5ITGAV
SCHEMBL6367900 0.87 ITGA4 (0.63) ITGB1ITGA4ITGB7ITGA5ITGAV

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1001764-A4 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO INC (US) 2005-08-24 EP claimed
US-6903075-B1 Heterocyclic amide compounds as cell adhesion inhibitors MERCK & CO., INC. (US) 2005-06-07 US claimed
JP-2002512625-A 2002-04-23 JP claimed
EP-1001764-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS Merck & Co., Inc. (a New Jersey corp.) (US) 2000-05-24 EP claimed
WO-1999064395-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO., INC. (US) 1999-12-16 WO claimed
WO-1998053814-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO., INC. (US) 1998-12-03 WO claimed