SCHEMBL5687544

SCHEMBL5687544

CCCCCCC1CCc2c(ccc3c2CCC(c2ccc(C#N)cc2)C3)C1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.43
CYP2C8 P10632 2/20 0.43
S1PR3 Q99500 2/20 0.43
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
S1PR1 P21453 7/20 0.38
S1PR4 O95977 1/20 0.38
S1PR5 Q9H228 1/20 0.38
GRM2 Q14416 1/20 0.37
SGPL1 O95470 3/20 0.37
TSHR P16473 1/20 0.36
HSD17B10 Q99714 1/20 0.36
DRD2 P14416 2/20 0.33
DRD3 P35462 2/20 0.33
HRH3 Q9Y5N1 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5687345 1.00 CYP3A4 (0.43) CYP3A4CYP2C8S1PR3CYP2D6CYP2C9
SCHEMBL5684665 0.99 CYP3A4 (0.41) CYP3A4CYP2C8S1PR3CYP2D6CYP2C9
SCHEMBL5686449 0.95 CYP3A4 (0.38) CYP3A4CYP2C8S1PR3CYP2D6CYP2C9
SCHEMBL5683979 0.91 MEN1 (0.34) CYP3A4CYP2C8S1PR3CYP2C9DRD2
SCHEMBL5684524 0.86 MCHR1 (0.34) DRD2DRD3HRH3
SCHEMBL14526395 0.84 GRM2 (0.38) CYP3A4CYP2C8S1PR3CYP2D6CYP2C9
SCHEMBL5684697 0.84 CYP3A4 (0.44) CYP3A4CYP2C8S1PR3CYP2D6CYP2C9
SCHEMBL5687011 0.84 CYP3A4 (0.44) CYP3A4CYP2C8S1PR3CYP2D6CYP2C9
SCHEMBL5683721 0.83 CYP3A4 (0.43) CYP3A4CYP2C8S1PR3CYP2D6CYP2C9
SCHEMBL5684309 0.79 CYP3A4 (0.39) CYP3A4CYP2C8S1PR3CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7067179-B1 Fused ring compound DAINIPPON INK AND CHEMICALS, INC. (JP) 2006-06-27 US disclosed
EP-1201632-B1 FUSED RING COMPOUND DAINIPPON INK & CHEMICALS (JP) 2006-03-29 EP disclosed
EP-1201632-A1 FUSED RING COMPOUND DAINIPPON INK AND CHEMICALS, INC. (JP) 2002-05-02 EP disclosed