SCHEMBL5683979

SCHEMBL5683979

CCCC1CCc2c(ccc3c2CCC(c2ccc(C#N)cc2)C3)C1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.34
MAPK1 P28482 1/20 0.34
KMT2A Q03164 1/20 0.34
HRH3 Q9Y5N1 2/20 0.34
ALDH1A1 P00352 2/20 0.34
MCHR1 Q99705 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C8 P10632 1/20 0.33
S1PR3 Q99500 1/20 0.33
CYP19A1 P11511 1/20 0.33
DRD2 P14416 1/20 0.33
DRD3 P35462 1/20 0.33
GRIA1 P42261 1/20 0.33
GRIA2 P42262 1/20 0.33
GRIA3 P42263 1/20 0.33
USP30 Q70CQ3 4/20 0.32
KCNH2 Q12809 1/20 0.32
LMNA P02545 1/20 0.32
MAPT P10636 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5686449 0.93 CYP3A4 (0.38) HRH3MCHR1CYP2C9CYP3A4CYP2C8
SCHEMBL5684665 0.92 CYP3A4 (0.41) HRH3CYP2C9CYP3A4CYP2C8S1PR3
SCHEMBL5687544 0.91 CYP3A4 (0.43) HRH3CYP2C9CYP3A4CYP2C8S1PR3
SCHEMBL5687345 0.91 CYP3A4 (0.43) HRH3CYP2C9CYP3A4CYP2C8S1PR3
SCHEMBL5684524 0.90 MCHR1 (0.34) HRH3MCHR1CYP19A1DRD2DRD3
SCHEMBL14526393 0.84 MEN1 (0.37) MEN1MAPK1KMT2AHRH3ALDH1A1
SCHEMBL5684932 0.83 CYP2C9 (0.35) MEN1MAPK1KMT2AALDH1A1CYP2C9
SCHEMBL5685243 0.83 DRD2 (0.44) MEN1MAPK1KMT2AALDH1A1MCHR1
SCHEMBL5684693 0.82 CYP3A4 (0.34) ALDH1A1CYP3A4CYP2C8S1PR3DRD2
SCHEMBL5684380 0.80 DRD2 (0.39) MEN1MAPK1KMT2AALDH1A1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7067179-B1 Fused ring compound DAINIPPON INK AND CHEMICALS, INC. (JP) 2006-06-27 US disclosed
EP-1201632-B1 FUSED RING COMPOUND DAINIPPON INK & CHEMICALS (JP) 2006-03-29 EP disclosed
EP-1201632-A1 FUSED RING COMPOUND DAINIPPON INK AND CHEMICALS, INC. (JP) 2002-05-02 EP disclosed