SCHEMBL5688807

SCHEMBL5688807

CNC(=O)c1cncc(-c2ccc(C(O)(c3c[nH]cn3)C(C)C)cc2)c1

nearest known ligand 0.56

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 14/20 0.56
CYP3A4 P08684 12/20 0.56
MKNK1 Q9BUB5 1/20 0.43
MKNK2 Q9HBH9 1/20 0.43
CDK7 P50613 1/20 0.43
XDH P47989 3/20 0.42
PIM1 P11309 1/20 0.41
PIM2 Q9P1W9 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5688304 0.87 CYP17A1 (0.68) CYP17A1CYP3A4
SCHEMBL5688557 0.82 CYP17A1 (0.51) CYP17A1CYP3A4
SCHEMBL5689340 0.80 CYP17A1 (0.47) CYP17A1CYP3A4PIM1PIM2
SCHEMBL5691318 0.79 CYP17A1 (0.58) CYP17A1CYP3A4
SCHEMBL7537438 0.79 CYP17A1 (0.65) CYP17A1CYP3A4
SCHEMBL7537443 0.79 CYP17A1 (0.65) CYP17A1CYP3A4
SCHEMBL4025212 0.79 CYP17A1 (0.65) CYP17A1CYP3A4
SCHEMBL4025340 0.79 CYP17A1 (0.65) CYP17A1CYP3A4
SCHEMBL5688423 0.79 CYP17A1 (0.46) CYP17A1CYP3A4
SCHEMBL5688992 0.78 CYP3A4 (0.56) CYP17A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1227086-B1 1-SUBSTITUTED PHENYL-1-(1H-IMIDAZOL-4-YL) ALCOHOLS, PROCESS FOR PRODUCING THE SAME AND USE THEREOF TAKEDA PHARMACEUTICAL (JP) 2006-03-29 EP disclosed
US-6518257-B1 1-substituted phenyl-1-(1h-imidazol-4-yl) alcohols, process for producing the same and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-02-11 US disclosed
EP-1227086-A1 1-SUBSTITUTED PHENYL-1-(1H-IMIDAZOL-4-YL) ALCOHOLS, PROCESS FOR PRODUCING THE SAME AND USE THEREOF Takeda Chemical Industries, Ltd. (JP) 2002-07-31 EP disclosed