SCHEMBL5688992

SCHEMBL5688992

CC(C)NC(=O)c1cccc(-c2ccc(C(O)(c3c[nH]cn3)C(C)C)cc2)c1

nearest known ligand 0.56

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 9/20 0.56
CYP17A1 P05093 7/20 0.56
NPSR1 Q6W5P4 1/20 0.46
ERN1 O75460 2/20 0.45
ROCK2 O75116 6/20 0.45
CYP3A5 P20815 2/20 0.43
PRKD1 Q15139 2/20 0.42
LIMK1 P53667 2/20 0.42
ROCK1 Q13464 2/20 0.41
RIPK1 Q13546 1/20 0.41
MAPK10 P53779 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5688304 0.91 CYP17A1 (0.68) CYP3A4CYP17A1
SCHEMBL5688568 0.88 CYP17A1 (0.53) CYP3A4CYP17A1ROCK2ROCK1
SCHEMBL5688798 0.88 CYP17A1 (0.54) CYP3A4CYP17A1CYP3A5RIPK1
SCHEMBL5691032 0.86 CYP17A1 (0.52) CYP3A4CYP17A1ROCK2ROCK1RIPK1
SCHEMBL5691318 0.83 CYP17A1 (0.58) CYP3A4CYP17A1
SCHEMBL4029239 0.82 CYP17A1 (0.66) CYP3A4CYP17A1NPSR1
SCHEMBL4025132 0.82 CYP17A1 (0.66) CYP3A4CYP17A1NPSR1
SCHEMBL7563594 0.81 CYP17A1 (0.66) CYP3A4CYP17A1
SCHEMBL5688564 0.81 CYP17A1 (0.66) CYP3A4CYP17A1
SCHEMBL5688705 0.81 CYP17A1 (0.44) CYP3A4CYP17A1ERN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1227086-B1 1-SUBSTITUTED PHENYL-1-(1H-IMIDAZOL-4-YL) ALCOHOLS, PROCESS FOR PRODUCING THE SAME AND USE THEREOF TAKEDA PHARMACEUTICAL (JP) 2006-03-29 EP disclosed
US-6518257-B1 1-substituted phenyl-1-(1h-imidazol-4-yl) alcohols, process for producing the same and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-02-11 US disclosed
EP-1227086-A1 1-SUBSTITUTED PHENYL-1-(1H-IMIDAZOL-4-YL) ALCOHOLS, PROCESS FOR PRODUCING THE SAME AND USE THEREOF Takeda Chemical Industries, Ltd. (JP) 2002-07-31 EP disclosed