SCHEMBL5688798

SCHEMBL5688798

CCNC(=O)c1cccc(-c2ccc(C(O)(c3c[nH]cn3)C(C)C)cc2)c1

nearest known ligand 0.54

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 12/20 0.54
CYP3A4 P08684 9/20 0.54
CDK8 P49336 1/20 0.46
CYP3A5 P20815 1/20 0.41
RIPK1 Q13546 1/20 0.40
MAPK1 P28482 1/20 0.40
AOC3 Q16853 2/20 0.38
ULK1 O75385 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5688304 0.89 CYP17A1 (0.68) CYP17A1CYP3A4CDK8
SCHEMBL5688992 0.88 CYP3A4 (0.56) CYP17A1CYP3A4CYP3A5RIPK1
SCHEMBL5688568 0.87 CYP17A1 (0.53) CYP17A1CYP3A4CDK8
SCHEMBL5691032 0.85 CYP17A1 (0.52) CYP17A1CYP3A4RIPK1
SCHEMBL4023743 0.83 CYP17A1 (0.67) CYP17A1CYP3A4RIPK1
SCHEMBL4024213 0.83 CYP17A1 (0.67) CYP17A1CYP3A4RIPK1
SCHEMBL5691318 0.82 CYP17A1 (0.58) CYP17A1CYP3A4CDK8
SCHEMBL5689203 0.82 CYP17A1 (0.45) CYP17A1CYP3A4ULK1
SCHEMBL5688634 0.81 CYP17A1 (0.52) CYP17A1CYP3A4
SCHEMBL5688411 0.80 CYP17A1 (0.47) CYP17A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1227086-B1 1-SUBSTITUTED PHENYL-1-(1H-IMIDAZOL-4-YL) ALCOHOLS, PROCESS FOR PRODUCING THE SAME AND USE THEREOF TAKEDA PHARMACEUTICAL (JP) 2006-03-29 EP disclosed
US-6518257-B1 1-substituted phenyl-1-(1h-imidazol-4-yl) alcohols, process for producing the same and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-02-11 US disclosed
EP-1227086-A1 1-SUBSTITUTED PHENYL-1-(1H-IMIDAZOL-4-YL) ALCOHOLS, PROCESS FOR PRODUCING THE SAME AND USE THEREOF Takeda Chemical Industries, Ltd. (JP) 2002-07-31 EP disclosed