SCHEMBL5688995

SCHEMBL5688995

CC(C)C(O)(c1cccc(-c2ccc(F)cc2)c1)c1cn(C(c2ccccc2)(c2ccccc2)c2ccccc2)cn1

nearest known ligand 0.52

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 6/20 0.52
CYP3A4 P08684 6/20 0.52
PTPN5 P54829 3/20 0.37
FLT3 P36888 1/20 0.35
PTPN1 P18031 2/20 0.34
ENPP2 Q13822 1/20 0.34
RORC P51449 1/20 0.34
SIRT2 Q8IXJ6 5/20 0.33
TNIK Q9UKE5 1/20 0.33
CLK1 P49759 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5691057 0.93 CYP17A1 (0.43) CYP17A1CYP3A4PTPN5PTPN1ENPP2
SCHEMBL5689004 0.91 CYP17A1 (0.44) CYP17A1CYP3A4ENPP2RORCSIRT2
SCHEMBL5688671 0.91 CYP17A1 (0.44) CYP17A1CYP3A4PTPN5PTPN1RORC
SCHEMBL5688405 0.90 CYP17A1 (0.46) CYP17A1CYP3A4PTPN5FLT3PTPN1
SCHEMBL5688756 0.89 CYP17A1 (0.52) CYP17A1CYP3A4PTPN5ENPP2RORC
SCHEMBL5688233 0.88 CYP3A4 (0.48) CYP17A1CYP3A4PTPN5ENPP2RORC
SCHEMBL5689153 0.88 CYP17A1 (0.39) CYP17A1CYP3A4ENPP2RORCSIRT2
SCHEMBL5688830 0.87 CYP17A1 (0.42) CYP17A1CYP3A4PTPN5PTPN1RORC
SCHEMBL5689382 0.87 CYP17A1 (0.43) CYP17A1CYP3A4PTPN5ENPP2RORC
SCHEMBL4025996 0.86 CYP3A4 (0.41) CYP17A1CYP3A4ENPP2RORCSIRT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1227086-B1 1-SUBSTITUTED PHENYL-1-(1H-IMIDAZOL-4-YL) ALCOHOLS, PROCESS FOR PRODUCING THE SAME AND USE THEREOF TAKEDA PHARMACEUTICAL (JP) 2006-03-29 EP disclosed
US-6518257-B1 1-substituted phenyl-1-(1h-imidazol-4-yl) alcohols, process for producing the same and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-02-11 US disclosed
EP-1227086-A1 1-SUBSTITUTED PHENYL-1-(1H-IMIDAZOL-4-YL) ALCOHOLS, PROCESS FOR PRODUCING THE SAME AND USE THEREOF Takeda Chemical Industries, Ltd. (JP) 2002-07-31 EP disclosed