SCHEMBL5689382

SCHEMBL5689382

CC(C)C(O)(c1cccc(-c2ccc(C#N)cc2)c1)c1cn(C(c2ccccc2)(c2ccccc2)c2ccccc2)cn1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 5/20 0.43
CYP3A4 P08684 5/20 0.43
ACSS2 Q9NR19 1/20 0.35
PTPN5 P54829 2/20 0.35
KAT6A Q92794 1/20 0.34
PSEN1 P49768 1/20 0.34
PSEN2 P49810 1/20 0.34
APH1B Q8WW43 1/20 0.34
NCSTN Q92542 1/20 0.34
APH1A Q96BI3 1/20 0.34
PSENEN Q9NZ42 1/20 0.34
MEN1 O00255 1/20 0.34
PHGDH O43175 1/20 0.33
ALDH1A3 P47895 1/20 0.33
PIN1 Q13526 1/20 0.33
FNTA P49354 1/20 0.33
FNTB P49356 1/20 0.33
RORC P51449 1/20 0.33
SYK P43405 1/20 0.33
ADAMTS4 O75173 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5688405 0.88 CYP17A1 (0.46) CYP17A1CYP3A4PTPN5RORCENPP2
SCHEMBL5688995 0.87 CYP17A1 (0.52) CYP17A1CYP3A4PTPN5RORCENPP2
SCHEMBL5688756 0.87 CYP17A1 (0.52) CYP17A1CYP3A4PTPN5RORCENPP2
SCHEMBL5688671 0.86 CYP17A1 (0.44) CYP17A1CYP3A4PTPN5RORC
SCHEMBL5688233 0.85 CYP3A4 (0.48) CYP17A1CYP3A4PTPN5RORCENPP2
SCHEMBL4032019 0.85 ACSS2 (0.38) CYP17A1CYP3A4ACSS2MEN1FNTA
SCHEMBL5691057 0.83 CYP17A1 (0.43) CYP17A1CYP3A4PTPN5RORCENPP2
SCHEMBL4025996 0.83 CYP3A4 (0.41) CYP17A1CYP3A4RORCENPP2
SCHEMBL5688830 0.82 CYP17A1 (0.42) CYP17A1CYP3A4PTPN5RORC
SCHEMBL5690498 0.82 CYP3A4 (0.47) CYP17A1CYP3A4RORCENPP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1227086-B1 1-SUBSTITUTED PHENYL-1-(1H-IMIDAZOL-4-YL) ALCOHOLS, PROCESS FOR PRODUCING THE SAME AND USE THEREOF TAKEDA PHARMACEUTICAL (JP) 2006-03-29 EP disclosed
US-6518257-B1 1-substituted phenyl-1-(1h-imidazol-4-yl) alcohols, process for producing the same and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-02-11 US disclosed
EP-1227086-A1 1-SUBSTITUTED PHENYL-1-(1H-IMIDAZOL-4-YL) ALCOHOLS, PROCESS FOR PRODUCING THE SAME AND USE THEREOF Takeda Chemical Industries, Ltd. (JP) 2002-07-31 EP disclosed