SCHEMBL5689052

SCHEMBL5689052

CC(=O)Nc1cc(-c2ccc(C(O)(c3cn(C(c4ccccc4)(c4ccccc4)c4ccccc4)cn3)C(C)C)cc2)cc(C(F)(F)F)c1

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 5/20 0.42
CYP17A1 P05093 4/20 0.42
NR2E1 Q9Y466 5/20 0.42
CYP2C19 P33261 2/20 0.40
ALDH1A1 P00352 1/20 0.40
CYP2C9 P11712 1/20 0.40
HPGD P15428 1/20 0.40
FYN P06241 1/20 0.39
P2RY14 Q15391 1/20 0.38
EGFR P00533 1/20 0.37
FGFR1 P11362 1/20 0.37
KDR P35968 1/20 0.37
IDH2 P48735 1/20 0.37
P2RX1 P51575 1/20 0.36
SYK P43405 1/20 0.36
MPO P05164 1/20 0.36
AURKA O14965 1/20 0.35
AURKB Q96GD4 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5688723 0.90 CYP17A1 (0.44) CYP3A4CYP17A1SYK
SCHEMBL5689005 0.88 CYP17A1 (0.55) CYP3A4CYP17A1FYNSYK
SCHEMBL5688259 0.88 CYP17A1 (0.50) CYP3A4CYP17A1CYP2C19ALDH1A1HPGD
SCHEMBL5690727 0.85 CYP17A1 (0.47) CYP3A4CYP17A1ALDH1A1FYNSYK
SCHEMBL5688662 0.83 CYP17A1 (0.40) CYP3A4CYP17A1CYP2C19ALDH1A1CYP2C9
SCHEMBL5688641 0.83 JAK2 (0.41) CYP3A4CYP17A1CYP2C19ALDH1A1HPGD
SCHEMBL5688707 0.82 CYP17A1 (0.40) CYP3A4CYP17A1
SCHEMBL5688671 0.81 CYP17A1 (0.44) CYP3A4CYP17A1ALDH1A1
SCHEMBL4030863 0.81 CYP17A1 (0.52) CYP3A4CYP17A1
SCHEMBL5691077 0.80 CYP17A1 (0.39) CYP3A4CYP17A1FYN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1227086-B1 1-SUBSTITUTED PHENYL-1-(1H-IMIDAZOL-4-YL) ALCOHOLS, PROCESS FOR PRODUCING THE SAME AND USE THEREOF TAKEDA PHARMACEUTICAL (JP) 2006-03-29 EP disclosed
US-6518257-B1 1-substituted phenyl-1-(1h-imidazol-4-yl) alcohols, process for producing the same and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-02-11 US disclosed
EP-1227086-A1 1-SUBSTITUTED PHENYL-1-(1H-IMIDAZOL-4-YL) ALCOHOLS, PROCESS FOR PRODUCING THE SAME AND USE THEREOF Takeda Chemical Industries, Ltd. (JP) 2002-07-31 EP disclosed