SCHEMBL5689182

SCHEMBL5689182

CC(C)C(O)(c1ccc(O)c(-c2ccc(F)cc2)c1)c1c[nH]cn1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 13/20 0.44
CYP3A4 P08684 11/20 0.44
CLK1 P49759 1/20 0.34
CLK2 P49760 1/20 0.34
DYRK1A Q13627 1/20 0.34
DYRK2 Q92630 1/20 0.34
CLK4 Q9HAZ1 1/20 0.34
DYRK1B Q9Y463 1/20 0.34
IDO1 P14902 2/20 0.33
NPC1 O15118 2/20 0.32
RAB9A P51151 2/20 0.32
MEN1 O00255 1/20 0.32
USP2 O75604 1/20 0.32
ALOX15 P16050 1/20 0.32
KMT2A Q03164 1/20 0.32
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5689193 0.86 CYP17A1 (0.42) CYP17A1CYP3A4CYP2C9CYP2C19
SCHEMBL5689007 0.85 CYP17A1 (0.58) CYP17A1CYP3A4RAB9AUSP2
SCHEMBL5689388 0.82 CYP17A1 (0.39) CYP17A1CYP3A4RAB9A
SCHEMBL5688562 0.82 BACE1 (0.39) CYP17A1CYP3A4CYP2C9CYP2C19
SCHEMBL5688515 0.81 CYP17A1 (0.63) CYP17A1CYP3A4
SCHEMBL5688390 0.76 CYP17A1 (0.47) CYP17A1CYP3A4
SCHEMBL5688934 0.75 CYP17A1 (0.52) CYP17A1CYP3A4IDO1
SCHEMBL5690835 0.74 CYP3A4 (0.41) CYP17A1CYP3A4CYP2C9CYP2C19
SCHEMBL5688522 0.74 CYP17A1 (0.57) CYP17A1CYP3A4CYP2C9
SCHEMBL5691085 0.74 CYP17A1 (0.37) CYP17A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1227086-B1 1-SUBSTITUTED PHENYL-1-(1H-IMIDAZOL-4-YL) ALCOHOLS, PROCESS FOR PRODUCING THE SAME AND USE THEREOF TAKEDA PHARMACEUTICAL (JP) 2006-03-29 EP disclosed
US-6518257-B1 1-substituted phenyl-1-(1h-imidazol-4-yl) alcohols, process for producing the same and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-02-11 US disclosed
EP-1227086-A1 1-SUBSTITUTED PHENYL-1-(1H-IMIDAZOL-4-YL) ALCOHOLS, PROCESS FOR PRODUCING THE SAME AND USE THEREOF Takeda Chemical Industries, Ltd. (JP) 2002-07-31 EP disclosed