SCHEMBL5689388

SCHEMBL5689388

CC(=O)Nc1ccc(C(O)(c2c[nH]cn2)C(C)C)cc1-c1ccc(F)cc1

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 10/20 0.39
CYP3A4 P08684 5/20 0.39
TOP2A P11388 2/20 0.37
RELA Q04206 1/20 0.36
CHRM3 P20309 1/20 0.36
RAB9A P51151 1/20 0.35
TDO2 P48775 1/20 0.35
NTRK1 P04629 1/20 0.33
ADORA3 P0DMS8 1/20 0.33
ADORA2A P29274 1/20 0.33
FYN P06241 1/20 0.33
FABP4 P15090 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5688562 0.82 BACE1 (0.39) CYP17A1CYP3A4
SCHEMBL5689182 0.82 CYP17A1 (0.44) CYP17A1CYP3A4RAB9A
SCHEMBL5688618 0.82 CYP17A1 (0.46) CYP17A1CYP3A4
SCHEMBL5690780 0.81 CYP17A1 (0.49) CYP17A1CYP3A4RAB9ATDO2
SCHEMBL5689193 0.80 CYP17A1 (0.42) CYP17A1CYP3A4
SCHEMBL5689007 0.79 CYP17A1 (0.58) CYP17A1CYP3A4RAB9A
SCHEMBL5688359 0.79 CYP17A1 (0.43) CYP17A1CYP3A4TOP2A
SCHEMBL5688374 0.78 CYP17A1 (0.63) CYP17A1CYP3A4
SCHEMBL5688476 0.77 CYP17A1 (0.34) CYP17A1CYP3A4TOP2ARELACHRM3
SCHEMBL7537711 0.76 CYP17A1 (0.64) CYP17A1CYP3A4RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1227086-B1 1-SUBSTITUTED PHENYL-1-(1H-IMIDAZOL-4-YL) ALCOHOLS, PROCESS FOR PRODUCING THE SAME AND USE THEREOF TAKEDA PHARMACEUTICAL (JP) 2006-03-29 EP disclosed
US-6518257-B1 1-substituted phenyl-1-(1h-imidazol-4-yl) alcohols, process for producing the same and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-02-11 US disclosed
EP-1227086-A1 1-SUBSTITUTED PHENYL-1-(1H-IMIDAZOL-4-YL) ALCOHOLS, PROCESS FOR PRODUCING THE SAME AND USE THEREOF Takeda Chemical Industries, Ltd. (JP) 2002-07-31 EP disclosed