SCHEMBL5689296

SCHEMBL5689296

CCCN1CCN(CCOc2ccc(Nc3ncc(C(N)=O)cn3)cc2F)CC1

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
AXL P30530 2/20 0.49
INSR P06213 1/20 0.49
CSF1R P07333 5/20 0.44
KDR P35968 4/20 0.44
EGFR P00533 6/20 0.43
LCK P06239 2/20 0.43
SRC P12931 1/20 0.43
BTK Q06187 2/20 0.42
MET P08581 1/20 0.41
P2RX3 P56373 1/20 0.41
TNK2 Q07912 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4507920 0.93 AXL (0.49) AXLINSRCSF1RKDREGFR
SCHEMBL4489929 0.91 AXL (0.57) AXLINSRCSF1RKDREGFR
SCHEMBL4499318 0.90 AXL (0.56) AXLINSRCSF1RKDREGFR
SCHEMBL5689284 0.90 AXL (0.47) AXLINSRCSF1RKDREGFR
SCHEMBL4495452 0.89 EGFR (0.48) AXLINSRCSF1RKDREGFR
SCHEMBL4500736 0.89 AXL (0.49) AXLINSRCSF1RKDREGFR
SCHEMBL5686178 0.89 CSF1R (0.52) AXLINSRCSF1RKDREGFR
SCHEMBL4480188 0.89 AXL (0.59) AXLINSRKDREGFRBTK
SCHEMBL4494805 0.86 AXL (0.52) AXLINSRCSF1RKDREGFR
SCHEMBL4495092 0.85 AXL (0.51) AXLINSRCSF1RKDREGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1648464-A1 2-AMINO-4-HYDROXY-5-PYRIMIDINCARBOXAMID DERIVATIVES AND RELATED COMPOUNDS AS T-CELL ACTIVATION INHIBITORS FOR THE TREATMENT OF INFLAMMATIONS AMGEN INC. (US) 2006-04-26 EP claimed
WO-2005009443-A1 2-AMINO-4-HYDROXY-5-PYRIMIDINECARBOXAMIDE DERIVATIVES AND RELATED COMPOUNDS AS INHIBITORS OF T CELL ACTIVATION FOR THE TREATMENT OF INFLAMMATORY DISEASES AMGEN INC. (US) 2005-02-03 WO claimed