SCHEMBL5689396

SCHEMBL5689396

COc1cccc(-c2ccc(C(O)(c3cn(C(c4ccccc4)(c4ccccc4)c4ccccc4)cn3)C(C)C)cc2)c1

nearest known ligand 0.43

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 6/20 0.43
CYP3A4 P08684 4/20 0.43
PTPN5 P54829 1/20 0.38
SIRT2 Q8IXJ6 7/20 0.37
TRPV1 Q8NER1 1/20 0.37
EGLN1 Q9GZT9 1/20 0.37
STIM1 Q13586 1/20 0.36
ORAI1 Q96D31 1/20 0.36
SLC13A5 Q86YT5 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5689096 0.87 CYP17A1 (0.50) CYP17A1CYP3A4SIRT2
SCHEMBL4025996 0.85 CYP3A4 (0.41) CYP17A1CYP3A4SIRT2
SCHEMBL5750734 0.85 CYP17A1 (0.48) CYP17A1CYP3A4SIRT2
SCHEMBL5688616 0.84 CYP17A1 (0.43) CYP17A1CYP3A4SIRT2
SCHEMBL5688671 0.84 CYP17A1 (0.44) CYP17A1CYP3A4PTPN5
SCHEMBL5688405 0.83 CYP17A1 (0.46) CYP17A1CYP3A4PTPN5SIRT2
SCHEMBL5688995 0.82 CYP17A1 (0.52) CYP17A1CYP3A4PTPN5SIRT2
SCHEMBL5688756 0.82 CYP17A1 (0.52) CYP17A1CYP3A4PTPN5SIRT2
SCHEMBL5688830 0.82 CYP17A1 (0.42) CYP17A1CYP3A4PTPN5
SCHEMBL5691363 0.82 CYP3A4 (0.46) CYP17A1CYP3A4SIRT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1227086-B1 1-SUBSTITUTED PHENYL-1-(1H-IMIDAZOL-4-YL) ALCOHOLS, PROCESS FOR PRODUCING THE SAME AND USE THEREOF TAKEDA PHARMACEUTICAL (JP) 2006-03-29 EP disclosed
US-6518257-B1 1-substituted phenyl-1-(1h-imidazol-4-yl) alcohols, process for producing the same and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-02-11 US disclosed
EP-1227086-A1 1-SUBSTITUTED PHENYL-1-(1H-IMIDAZOL-4-YL) ALCOHOLS, PROCESS FOR PRODUCING THE SAME AND USE THEREOF Takeda Chemical Industries, Ltd. (JP) 2002-07-31 EP disclosed