SCHEMBL5690498

SCHEMBL5690498

CC(C)C(O)(c1cccc(-c2cccnc2)c1)c1cn(C(c2ccccc2)(c2ccccc2)c2ccccc2)cn1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 8/20 0.47
CYP17A1 P05093 5/20 0.47
RORC P51449 2/20 0.38
SIRT2 Q8IXJ6 1/20 0.36
ENPP2 Q13822 1/20 0.36
CYP2E1 P05181 3/20 0.36
CYP2A6 P11509 3/20 0.36
CYP2C9 P11712 3/20 0.36
CYP2B6 P20813 3/20 0.36
CYP2C19 P33261 3/20 0.36
KMO O15229 1/20 0.36
KCNA5 P22460 4/20 0.35
MC4R P32245 1/20 0.35
CYP2D6 P10635 1/20 0.34
KDR P35968 1/20 0.34
KCNH2 Q12809 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5688233 0.89 CYP3A4 (0.48) CYP3A4CYP17A1RORCSIRT2ENPP2
SCHEMBL5691057 0.85 CYP17A1 (0.43) CYP3A4CYP17A1RORCSIRT2ENPP2
SCHEMBL5688405 0.85 CYP17A1 (0.46) CYP3A4CYP17A1RORCSIRT2ENPP2
SCHEMBL5689298 0.84 CYP17A1 (0.43) CYP3A4CYP17A1RORCSIRT2ENPP2
SCHEMBL5688756 0.84 CYP17A1 (0.52) CYP3A4CYP17A1RORCSIRT2ENPP2
SCHEMBL5688995 0.84 CYP17A1 (0.52) CYP3A4CYP17A1RORCSIRT2ENPP2
SCHEMBL5688671 0.83 CYP17A1 (0.44) CYP3A4CYP17A1RORC
SCHEMBL5688642 0.82 CYP17A1 (0.41) CYP3A4CYP17A1RORCSIRT2ENPP2
SCHEMBL5688980 0.82 CYP17A1 (0.41) CYP3A4CYP17A1RORCSIRT2ENPP2
SCHEMBL5688667 0.82 CYP17A1 (0.40) CYP3A4CYP17A1RORCSIRT2ENPP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1227086-B1 1-SUBSTITUTED PHENYL-1-(1H-IMIDAZOL-4-YL) ALCOHOLS, PROCESS FOR PRODUCING THE SAME AND USE THEREOF TAKEDA PHARMACEUTICAL (JP) 2006-03-29 EP disclosed
US-6518257-B1 1-substituted phenyl-1-(1h-imidazol-4-yl) alcohols, process for producing the same and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-02-11 US disclosed
EP-1227086-A1 1-SUBSTITUTED PHENYL-1-(1H-IMIDAZOL-4-YL) ALCOHOLS, PROCESS FOR PRODUCING THE SAME AND USE THEREOF Takeda Chemical Industries, Ltd. (JP) 2002-07-31 EP disclosed