SCHEMBL5690780

SCHEMBL5690780

CC(=O)Nc1ccc(F)c(-c2ccc(C(O)(c3c[nH]cn3)C(C)C)cc2)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 11/20 0.49
CYP3A4 P08684 5/20 0.49
IDO1 P14902 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.38
CPT1A P50416 1/20 0.36
DDR2 Q16832 1/20 0.35
CLK1 P49759 1/20 0.35
DYRK1A Q13627 1/20 0.35
DYRK2 Q92630 1/20 0.35
DYRK1B Q9Y463 1/20 0.35
RORC P51449 1/20 0.35
KIF11 P52732 1/20 0.35
TDO2 P48775 1/20 0.35
MEN1 O00255 1/20 0.34
NPC1 O15118 1/20 0.34
ALDH1A1 P00352 1/20 0.34
MAPT P10636 1/20 0.34
MAOA P21397 1/20 0.34
RAB9A P51151 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5688374 0.87 CYP17A1 (0.63) CYP17A1CYP3A4SMN1; SMN2
SCHEMBL5689213 0.86 CYP17A1 (0.48) CYP17A1CYP3A4IDO1DDR2TDO2
SCHEMBL5688618 0.85 CYP17A1 (0.46) CYP17A1CYP3A4CPT1A
SCHEMBL5689340 0.83 CYP17A1 (0.47) CYP17A1CYP3A4RORC
SCHEMBL29478298 0.82 CYP17A1 (0.66) CYP17A1CYP3A4
SCHEMBL5688564 0.82 CYP17A1 (0.66) CYP17A1CYP3A4
SCHEMBL7563594 0.82 CYP17A1 (0.66) CYP17A1CYP3A4
SCHEMBL5689065 0.82 CYP17A1 (0.48) CYP17A1CYP3A4DYRK1AMEN1ALDH1A1
SCHEMBL5690714 0.81 CYP17A1 (0.49) CYP17A1CYP3A4KIF11
SCHEMBL5689388 0.81 CYP17A1 (0.39) CYP17A1CYP3A4TDO2RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1227086-B1 1-SUBSTITUTED PHENYL-1-(1H-IMIDAZOL-4-YL) ALCOHOLS, PROCESS FOR PRODUCING THE SAME AND USE THEREOF TAKEDA PHARMACEUTICAL (JP) 2006-03-29 EP disclosed
US-6518257-B1 1-substituted phenyl-1-(1h-imidazol-4-yl) alcohols, process for producing the same and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-02-11 US disclosed
EP-1227086-A1 1-SUBSTITUTED PHENYL-1-(1H-IMIDAZOL-4-YL) ALCOHOLS, PROCESS FOR PRODUCING THE SAME AND USE THEREOF Takeda Chemical Industries, Ltd. (JP) 2002-07-31 EP disclosed