SCHEMBL5690967

SCHEMBL5690967

c1ccc2c(c1)CCC2NC1CCNCC1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDPK1 O15530 1/20 0.54
KDM1A O60341 7/20 0.51
MAOA P21397 4/20 0.51
MAOB P27338 4/20 0.51
SLC18A3 Q16572 1/20 0.51
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
BCHE P06276 1/20 0.46
ADRA2B P18089 1/20 0.46
ADRA2C P18825 1/20 0.46
ACHE P22303 1/20 0.46
ADRA1A P35348 1/20 0.46
HTR6 P50406 1/20 0.46
HTR2C P28335 2/20 0.46
CISD1 Q9NZ45 1/20 0.44
SLC6A2 P23975 1/20 0.44
HTR1B P28222 1/20 0.44
HTR2A P28223 1/20 0.44
SLC6A4 P31645 1/20 0.44
FADS1 O60427 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5690934 0.94 SLC18A3 (0.50) PDPK1KDM1AMAOAMAOBSLC18A3
SCHEMBL20608227 0.83 SLC18A3 (0.62) PDPK1KDM1AMAOAMAOBSLC18A3
SCHEMBL20321172 0.83 SLC18A3 (0.62) PDPK1KDM1AMAOAMAOBSLC18A3
SCHEMBL20608209 0.83 SLC18A3 (0.62) PDPK1KDM1AMAOAMAOBSLC18A3
SCHEMBL2322457 0.82 PDPK1 (0.70) PDPK1KDM1AMAOAMAOBSLC18A3
Hydrochloric Acid SCHEMBL7123292 0.80 PDPK1 (0.68) PDPK1KDM1AMAOAMAOBSLC18A3
SCHEMBL4209025 0.79 PDPK1 (0.57) PDPK1KDM1AMAOAMAOBSLC18A3
SCHEMBL12431685 0.78 SLC18A3 (0.52) PDPK1KDM1AMAOAMAOBSLC18A3
SCHEMBL3853169 0.76 HTR2C (0.53) CA1CA2HTR6HTR2C
SCHEMBL3316700 0.75 EPHX1 (0.50) PDPK1SLC18A3ADRA2BADRA2CADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1658269-A1 FUSED COMPOUNDS THAT INHIBIT VANILLOID RECEPTOR SUBTYPE 1 (VR1) RECEPTOR Abbott Laboratories (US) 2006-05-24 EP disclosed
WO-2004111009-A1 FUSED COMPOUNDS THAT INHIBIT VANILLOID RECEPTOR SUBTYPE 1 (VR1) RECEPTOR ABBOTT LABORATORIES (US) 2004-12-23 WO disclosed