SCHEMBL569174

SCHEMBL569174

O=C1CCOc2cc(F)ccc21

nearest known ligand 0.64

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAOB P27338 17/20 0.64
MAOA P21397 1/20 0.64
GRM5 P41594 6/20 0.61
NPC1 O15118 1/20 0.49
ALDH1A1 P00352 1/20 0.49
HPGD P15428 1/20 0.49
NFKB1 P19838 1/20 0.49
RAB9A P51151 1/20 0.49
NFKB2 Q00653 1/20 0.49
RELA Q04206 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29758920 1.00 MAOB (0.64) MAOBMAOAGRM5NPC1ALDH1A1
Hydrochloric Acid SCHEMBL27916588 0.98 MAOB (0.62) MAOBMAOAGRM5NPC1ALDH1A1
SCHEMBL915230 0.89 MAOB (0.51) MAOBMAOAGRM5NPC1ALDH1A1
SCHEMBL15818326 0.86 MAOB (0.59) MAOBMAOAGRM5NPC1ALDH1A1
SCHEMBL769330 0.85 FABP6 (0.58) MAOBMAOAGRM5NPC1ALDH1A1
SCHEMBL15818861 0.82 MAOB (0.58) MAOBMAOAGRM5NPC1ALDH1A1
SCHEMBL1924055 0.81 MAOB (0.54) MAOBMAOAGRM5NPC1RAB9A
SCHEMBL4728838 0.79 MAOB (0.66) MAOBMAOAGRM5NPC1ALDH1A1
SCHEMBL2961997 0.78 MAOB (0.54) MAOBMAOAGRM5NPC1ALDH1A1
SCHEMBL8578811 0.78 MAOB (0.64) MAOBMAOAGRM5NPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 222 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112079826-B Steroid synthetase inhibitor and treatment application thereof 广州中医药大学(广州中医药研究院) 2022-07-29 CN claimed
WO-2022057142-A1 STEROID SYNTHETASE INHIBITORS AND THERAPEUTIC USE THEREOF 广州中医药大学(广州中医药研究院) 2022-03-24 WO claimed
CN-112079826-A Steroid synthetase inhibitor and treatment application thereof 广州中医药大学(广州中医药研究院) 2020-12-15 CN claimed
US-12497377-B2 Tricyclic spiro compound ONO PHARMACEUTICAL CO., LTD. (JP) 2025-12-16 US disclosed
WO-2025036382-A1 SULFONAMIDE COMPOUND, AND PREPARATION METHOD THEREFOR AND USE THEREOF 上海复宏汉霖生物医药有限公司 2025-02-20 WO disclosed
US-12157726-B2 P-phenylenediamine derivative as potassium channel regulator and preparation method and medical application thereof SHANGHAI ZHIMENG BIOPHARMA INC. 2024-12-03 US disclosed
US-20240368109-A1 ALLOSTERIC MODULATORS OF NICOTINIC ACETYLCHOLINE RECEPTORS MERCK SHARP & DOHME LLC (US) 2024-11-07 US disclosed
EP-4404935-A1 ALLOSTERIC MODULATORS OF NICOTINIC ACETYLCHOLINE RECEPTORS Merck Sharp & Dohme LLC (US) 2024-07-31 EP disclosed
WO-2024140431-A1 COMPOUNDS COMPRISING HETEROARYL RINGS AND COMPOSITIONS AND METHODS THEREOF IONGEN THERAPEUTICS CO., LTD. (CN) 2024-07-04 WO disclosed
US-20240182436-A1 SUBSTITUTED SULFONAMIDE-CHROMAN COMPOUNDS, AND PHARMACEUTICAL COMPOSITIONS, AND METHODS OF USE THEREOF SUMITOMO PHARMA AMERICA, INC. (US) 2024-06-06 US disclosed
WO-2024040267-A2 DIRECT SYNTHESIS OF N-(3-SUBSTITUTED-CHROMAN-4-YL)-7H- PYRROLO[2,3-D]PYRIMIDIN-4-AMINES AND DERIVATIVES THEREOF MITOKININ, INC. (US) 2024-02-22 WO disclosed
US-6316437-B1 ADRENERGIC RECEPTOR ANTAGONISTS MERCK & CO., INC. 2001-11-13 US disclosed
WO-2001045704-A1 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE MERCK & CO., INC. (US) 2001-06-28 WO disclosed
WO-1998009969-A1 NOVEL ARYL-PYRIDAZINES ASTRA PHARMACEUTICALS LTD. (GB) 1998-03-12 WO disclosed
US-5521147-A HERBICIDES FMC CORPORATION (US) 1996-05-28 US disclosed
US-4992564-A Preparation of 6-substituted 4-chromanones MALLINCKRODT, INC. (US) 1991-02-12 US disclosed
EP-0400403-A2 N-aryl-nitrogen-heterocycles BAYER AG (DE) 1990-12-05 EP disclosed
US-4918203-A Preparation of 6-substituted 4-chromanones MALLINCKRODT INC. 1990-04-17 US disclosed
EP-0228172-B1 PREPARATION OF 6-SUBSTITUTED 4-CHROMANONES Mallinckrodt, Inc. (a Delaware corporation) (US) 1990-03-07 EP disclosed
EP-0228172-A1 Preparation of 6-substituted 4-chromanones Mallinckrodt, Inc. (a Delaware corporation) (US) 1987-07-08 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12157726-B2 P-phenylenediamine derivative as potassium channel regulator and preparation method and medical application thereof KCNJ2, KCNN2, KCNH2 MAOB 1320/4885MAOA 1302/4885GRM5 1632/4885
US-20240368109-A1 ALLOSTERIC MODULATORS OF NICOTINIC ACETYLCHOLINE RECEPTORS CHRNA7, CHRNA5, CHRNA6 MAOB 386/4885MAOA 294/4885GRM5 93/4885
US-12497377-B2 Tricyclic spiro compound PTGER4, PTGER1, PTGER3 MAOB 2126/4885MAOA 2145/4885GRM5 874/4885
US-20240182436-A1 SUBSTITUTED SULFONAMIDE-CHROMAN COMPOUNDS, AND PHARMACEUTICAL COMPOSITIONS, AND METHODS OF USE THEREOF ARSA, SNCA, F12 MAOB 186/4885MAOA 267/4885GRM5 1572/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.