SCHEMBL5693144

SCHEMBL5693144

OC1c2ccccc2CN1Cc1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 7/20 0.48
GRIN1 Q05586 1/20 0.48
GRIN2B Q13224 1/20 0.48
MAPT P10636 1/20 0.44
FUCA1 P04066 2/20 0.42
GBA1 P04062 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29760303 1.00 SIGMAR1 (0.48) SIGMAR1GRIN1GRIN2BMAPTFUCA1
SCHEMBL17231981 0.84 SIGMAR1 (0.49) SIGMAR1
SCHEMBL29774325 0.83 GAA (0.47) SIGMAR1GRIN1GRIN2BGBA1
SCHEMBL13978050 0.80 GBA1 (0.43) SIGMAR1GRIN1GRIN2BGBA1
SCHEMBL24755096 0.79 HDAC1 (0.39)
SCHEMBL7044789 0.79 ACE (0.52) SIGMAR1GRIN1GRIN2B
SCHEMBL7044790 0.79 ACE (0.52) SIGMAR1GRIN1GRIN2B
SCHEMBL7044785 0.79 ACE (0.52) SIGMAR1GRIN1GRIN2B
SCHEMBL14012100 0.79 PRCP (0.49) MAPT
SCHEMBL13079294 0.77 SIGMAR1 (0.42) SIGMAR1GRIN1GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1528923-B1 N-((3-OXO-2,3-DIHYDRO-1H-ISOINDOL-1-YL)ACETYL)GUANIDINE DERIVATIVES AS NHE1-INHIBITORS FOR THE TREATMENT OF INFARCTION AND ANGINA PECTORIS SANOFI AVENTIS DEUTSCHLAND (DE) 2006-05-03 EP disclosed