Arimoclomol

Arimoclomol

SCHEMBL5699321

O=C(O[C@@H](C(=O)O)[C@@H](OC(=O)c1ccccc1)C(=O)O)c1ccccc1.[O-][n+]1cccc(C(Cl)=NOC[C@H](O)CN2CCCCC2)c1

nearest known ligand 0.47

Full drug profile on Sugi Atlas →

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HSF1 Q00613 13/20 0.47
ABCB1 P08183 5/20 0.42
MAPK1 P28482 1/20 0.41
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Arimoclomol SCHEMBL2324741 0.88 HSF1 (0.54) HSF1ABCB1
Arimoclomol SCHEMBL1896428 0.88 HSF1 (0.54) HSF1ABCB1
Arimoclomol SCHEMBL12254223 0.88 HSF1 (0.54) HSF1ABCB1
Arimoclomol SCHEMBL25257807 0.88 HSF1 (0.54) HSF1ABCB1
Arimoclomol SCHEMBL12254225 0.88 HSF1 (0.54) HSF1ABCB1
Arimoclomol SCHEMBL25258754 0.88 HSF1 (0.54) HSF1ABCB1
Arimoclomol SCHEMBL196123 0.88 HSF1 (0.54) HSF1ABCB1
Arimoclomol SCHEMBL5699241 0.88 HSF1 (0.54) HSF1ABCB1
Arimoclomol SCHEMBL7052423 0.87 HSF1 (0.53) HSF1ABCB1
Arimoclomol SCHEMBL5699253 0.87 HSF1 (0.53) HSF1ABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7126002-B2 Pyridine-1-oxide derivative, and process for its transformation into pharmaceutically effective compounds CYTRX CORPORATION (US) 2006-10-24 US disclosed
EP-1274685-B1 A PYRIDINE-N-OXIDE DERIVATIVE, AND PROCESS FOR ITS TRANSFORMATION INTO PHARMACEUTICALLY EFFECTIVE COMPOUNDS BIOREX KUTATO FEJLESZTOE KFT (HU) 2006-07-12 EP disclosed
US-20040006232-A1 Pyridine-1-oxide derivative, and process for its transformation into pharmaceutically effective compounds KEMPHARM, INC. 2004-01-08 US disclosed
EP-1274685-A1 A PYRIDINE-1-OXIDE DERIVATIVE, AND PROCESS FOR ITS TRANSFORMATION INTO PHARMACEUTICALLY EFFECTIVE COMPOUNDS BIOREX KUTATO ES FEJLESZTÖ RT. (HU) 2003-01-15 EP disclosed
WO-2001079174-A1 A PYRIDINE-1-OXIDE DERIVATIVE, AND PROCESS FOR ITS TRANSFORMATION INTO PHARMACEUTICALLY EFFECTIVE COMPOUNDS BIOREX Kutató és Fejlesztő Rt. (HU) 2001-10-25 WO disclosed