SCHEMBL5700903

SCHEMBL5700903

COC(=O)C[C@@H](NC(=O)c1ccc(OC)c(OC)c1)c1ccc(NC(=O)Cc2ccc(NC(=O)Nc3ccccc3C)c(OC)c2)cc1

nearest known ligand 0.64

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 12/20 0.64
ITGA4 P13612 12/20 0.64
EPHX2 P34913 1/20 0.47
P2RX7 Q99572 1/20 0.46
ITGB7 P26010 1/20 0.45
BCHE P06276 2/20 0.45
ACHE P22303 2/20 0.45
ROCK2 O75116 1/20 0.44
ROCK1 Q13464 1/20 0.44
MAPT P10636 2/20 0.44
KMT2A Q03164 2/20 0.44
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 1/20 0.44
HPGD P15428 1/20 0.44
MEN1 O00255 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5700909 1.00 ITGB1 (0.64) ITGB1ITGA4EPHX2P2RX7ITGB7
SCHEMBL5700856 0.94 ITGB1 (0.71) ITGB1ITGA4EPHX2P2RX7ITGB7
SCHEMBL5700846 0.94 ITGB1 (0.71) ITGB1ITGA4EPHX2P2RX7ITGB7
SCHEMBL5700827 0.93 ITGB1 (0.70) ITGB1ITGA4ITGB7KMT2AMEN1
SCHEMBL5700821 0.93 ITGB1 (0.70) ITGB1ITGA4ITGB7KMT2AMEN1
SCHEMBL5700956 0.92 ITGB1 (0.64) ITGB1ITGA4ITGB7MAPTKMT2A
SCHEMBL5700962 0.92 ITGB1 (0.64) ITGB1ITGA4ITGB7MAPTKMT2A
SCHEMBL5700904 0.89 ITGB1 (0.70) ITGB1ITGA4EPHX2P2RX7ITGB7
SCHEMBL5700900 0.89 ITGB1 (0.70) ITGB1ITGA4EPHX2P2RX7ITGB7
SCHEMBL5700873 0.88 ITGB1 (0.61) ITGB1ITGA4ITGB7ROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1027328-B1 SUBSTITUTED ANILIDES AVENTIS PHARMA LTD (GB) 2006-08-23 EP disclosed
US-6479519-B1 INHIBITORS OF CELL ADHESION; TREATMENT OF ASTHMA OR INFLAMMATORY BOWEL DISEASE AVENTIS PHARMA LIMITED (GB) 2002-11-12 US disclosed