SCHEMBL5703530

SCHEMBL5703530

Nc1ccc(CNCc2ccc3ccccc3c2)cc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MC5R P33032 5/20 0.64
MC4R P32245 3/20 0.64
MC3R P41968 3/20 0.60
ROCK1 Q13464 2/20 0.59
MAPK1 P28482 1/20 0.58
ALDH1A1 P00352 2/20 0.52
CYP3A4 P08684 2/20 0.52
HSD17B10 Q99714 2/20 0.52
MC1R Q01726 2/20 0.51
CA12 O43570 1/20 0.50
CA1 P00915 1/20 0.50
CA2 P00918 1/20 0.50
CA4 P22748 1/20 0.50
CYP1A2 P05177 1/20 0.47
CYP2A6 P11509 1/20 0.47
HDAC3 O15379 1/20 0.46
HDAC1 Q13547 1/20 0.46
HDAC2 Q92769 1/20 0.46
HDAC8 Q9BY41 1/20 0.46
ALOX15 P16050 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6008141 0.88 MC5R (0.71) MC5RMC4RMC3RROCK1MAPK1
SCHEMBL4017226 0.86 MC5R (0.65) MC5RMC4RMC3RROCK1MAPK1
SCHEMBL7250915 0.85 MC5R (0.69) MC5RMC4RMC3RROCK1MAPK1
Hydrochloric Acid SCHEMBL31120720 0.85 MC5R (0.62) MC5RMC4RMC3RROCK1MAPK1
Hydrochloric Acid SCHEMBL31120721 0.85 MC5R (0.62) MC5RMC4RMC3RROCK1MAPK1
SCHEMBL5703579 0.81 MC5R (0.59) MC5RMC4RMC3RROCK1MAPK1
SCHEMBL27502280 0.81 MC5R (0.59) MC5RMC4RMC3RROCK1MAPK1
Hydrochloric Acid SCHEMBL6417210 0.80 MC5R (0.57) MC5RMC4RMC3RROCK1MAPK1
SCHEMBL2125786 0.79 TDP1 (0.55) ALDH1A1CYP3A4CA12CA1CA2
SCHEMBL8826336 0.79 KDM4E (0.63) MC5RMC4RMC3RROCK1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1514112-B1 METHOD FOR IDENTIFYING AN ALLOSTERIC EFFECTOR OF A RECEPTOR CENTRE NAT RECH SCIENT (FR) 2006-09-06 EP disclosed
US-20060194259-A1 Method for isolating an allosteric effector of a receptor UNIVERSITE LOUIS PASTEUR DE STRASSOURG (FR) 2006-08-31 US disclosed