SCHEMBL5705606

SCHEMBL5705606

CN1c2ccccc2C(C(O)=S)c2ccccc21

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 1/20 0.56
HDAC7 Q8WUI4 1/20 0.56
HDAC5 Q9UQL6 1/20 0.56
EGFR P00533 2/20 0.50
SRC P12931 1/20 0.50
CHEK1 O14757 1/20 0.43
AURKA O14965 1/20 0.43
DAPK3 O43293 1/20 0.43
JAK2 O60674 1/20 0.43
PRKD3 O94806 1/20 0.43
MAP4K4 O95819 1/20 0.43
PAK4 O96013 1/20 0.43
ABL1 P00519 1/20 0.43
NTRK1 P04629 1/20 0.43
LCK P06239 1/20 0.43
FYN P06241 1/20 0.43
CSF1R P07333 1/20 0.43
RET P07949 1/20 0.43
IGF1R P08069 1/20 0.43
MET P08581 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Chlorobenzene SCHEMBL28307149 0.91 HDAC4 (0.49) HDAC4HDAC7HDAC5EGFRSRC
SCHEMBL7755161 0.83 HDAC4 (0.42) HDAC4HDAC7HDAC5EGFRSRC
SCHEMBL8331436 0.81 HDAC4 (0.43) HDAC4HDAC7HDAC5EGFRSRC
SCHEMBL7752463 0.81 HDAC4 (0.43) HDAC4HDAC7HDAC5EGFRSRC
SCHEMBL2989515 0.80 HDAC4 (0.66) HDAC4HDAC7HDAC5EGFRSRC
SCHEMBL31613807 0.80 HDAC4 (0.66) HDAC4HDAC7HDAC5EGFRSRC
SCHEMBL5161928 0.79 HDAC4 (0.47) HDAC4HDAC7HDAC5EGFRSRC
Hydrochloric Acid SCHEMBL2982836 0.78 HDAC4 (0.64) HDAC4HDAC7HDAC5EGFRSRC
SCHEMBL8331385 0.78 HDAC4 (0.50) HDAC4HDAC7HDAC5EGFRSRC
SCHEMBL7756492 0.78 HDAC4 (0.40) HDAC4HDAC7HDAC5EGFRSRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 33 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106749404-B A kind of preparation method generating chemiluminescent compound with alkaline phosphatase enzyme reaction 湖南远璟生物技术有限公司 2019-01-04 CN claimed
CN-106749404-A A kind of preparation method with the alkaline phosphatase enzyme reaction chemiluminescent compound of generation 湖南远璟生物技术有限公司 2017-05-31 CN claimed
EP-0755457-B1 Novel Aryl-N-Alkylacridanthiocarboxylate derivatives useful for chemiluminescent detection LUMIGEN INC (US) 2001-02-21 EP claimed
EP-0755457-A4 NOVEL ARYL-N-ALKYLACRIDANTHIOCARBOXYLATE DERIVATIVES USEFUL FOR CHEMILUMINESCENT DETECTION LUMIGEN INC (US) 1997-07-16 EP claimed
EP-0755457-A1 NOVEL ARYL-N-ALKYLACRIDANTHIOCARBOXYLATE DERIVATIVES USEFUL FOR CHEMILUMINESCENT DETECTION LUMIGEN, INC. (US) 1997-01-29 EP claimed
WO-1995028495-A1 NOVEL ARYL-N-ALKYLACRIDANTHIOCARBOXYLATE DERIVATIVES USEFUL FOR CHEMILUMINESCENT DETECTION LUMIGEN, INC. (US) 1995-10-26 WO claimed
CN-106749404-B A kind of preparation method generating chemiluminescent compound with alkaline phosphatase enzyme reaction 湖南远璟生物技术有限公司 2019-01-04 CN disclosed
CN-106749404-B A kind of preparation method generating chemiluminescent compound with alkaline phosphatase enzyme reaction 湖南远璟生物技术有限公司 2019-01-04 CN disclosed
CN-106749404-A A kind of preparation method with the alkaline phosphatase enzyme reaction chemiluminescent compound of generation 湖南远璟生物技术有限公司 2017-05-31 CN disclosed
EP-1054933-B1 CHEMILUMINESCENT REACTIONS USING DIHYDROXYAROMATIC COMPOUNDS AND HETEROCYCLIC ENOL PHOSPHATES LUMIGEN INC (US) 2006-09-06 EP disclosed
CN-1173954-C Compounds, compositions and methods for generating chemiluminescence by reaction with phosphatases 3 2004-11-03 CN disclosed
US-6635437-B2 Useful in methods for producing light and in assays for phosphatase enzymes and enzyme inhibitors and in assays employing enzyme-labeled specific binding pairs LUMIGEN, INC. 2003-10-21 US disclosed
EP-1054933-A4 CHEMILUMINESCENT REACTIONS USING DIHYDROXYAROMATIC COMPOUNDS AND HETEROCYCLIC ENOL PHOSPHATES LUMIGEN INC (US) 2003-07-09 EP disclosed
US-5772926-A ANALYSIS OF HYDROLYTIC ENZYMES AND ENZYME INHIBITORS; LABELED BINDING PAIRS LUMIGEN, INC. (US) 1998-06-30 US disclosed
CN-1180349-A Compounds, compositions and methods for generating chemiluminescence by reaction with phosphatases LUMIGEN INC (US) 1998-04-29 CN disclosed
EP-0819119-A1 COMPOUNDS, COMPOSITIONS AND METHODS FOR GENERATING CHEMILUMINESCENCE WITH PHOSPHATASE ENZYMES LUMIGEN, INC. (US) 1998-01-21 EP disclosed
WO-1997026245-A1 COMPOUNDS, COMPOSITIONS AND METHODS FOR GENERATING CHEMILUMINESCENCE WITH PHOSPHATASE ENZYMES LUMIGEN, INC. (US) 1997-07-24 WO disclosed
EP-0755457-A4 NOVEL ARYL-N-ALKYLACRIDANTHIOCARBOXYLATE DERIVATIVES USEFUL FOR CHEMILUMINESCENT DETECTION LUMIGEN INC (US) 1997-07-16 EP disclosed
EP-0755457-A1 NOVEL ARYL-N-ALKYLACRIDANTHIOCARBOXYLATE DERIVATIVES USEFUL FOR CHEMILUMINESCENT DETECTION LUMIGEN, INC. (US) 1997-01-29 EP disclosed
WO-1995028495-A1 NOVEL ARYL-N-ALKYLACRIDANTHIOCARBOXYLATE DERIVATIVES USEFUL FOR CHEMILUMINESCENT DETECTION LUMIGEN, INC. (US) 1995-10-26 WO disclosed