SCHEMBL5707229

SCHEMBL5707229

Cc1ccc(C(=O)Nc2ccc3[nH]ncc3c2)cc1F

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 6/20 0.72
RAB9A P51151 6/20 0.72
MAOB P27338 4/20 0.68
ROCK2 O75116 2/20 0.67
MAP4K4 O95819 2/20 0.67
RPS6KB1 P23443 2/20 0.67
CLK2 P49760 2/20 0.67
ROCK1 Q13464 2/20 0.67
DYRK1A Q13627 2/20 0.67
CLK4 Q9HAZ1 2/20 0.67
DYRK3 O43781 1/20 0.67
CSNK2A1 P68400 1/20 0.67
MKNK2 Q9HBH9 1/20 0.67
PRKD3 O94806 1/20 0.65
PRKG1 Q13976 1/20 0.65
PRKD2 Q9BZL6 1/20 0.65
SGK2 Q9HBY8 1/20 0.65
STK17A Q9UEE5 1/20 0.65
JAK2 O60674 1/20 0.64
MEN1 O00255 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15764665 0.89 MAOB (0.70) NPC1RAB9AMAOBROCK2MAP4K4
SCHEMBL5415117 0.86 MAOB (0.80) NPC1RAB9AMAOBROCK2MAP4K4
SCHEMBL15887002 0.84 MAOB (0.81) NPC1RAB9AMAOBROCK2MAP4K4
SCHEMBL1664461 0.84 NPC1 (1.00) NPC1RAB9AMAOBROCK2MAP4K4
SCHEMBL5415932 0.81 MAOB (0.69) NPC1RAB9AMAOBROCK2MAP4K4
SCHEMBL5414918 0.81 NPC1 (0.85) NPC1RAB9AMAOBROCK2MAP4K4
SCHEMBL15886999 0.81 MAOB (0.83) NPC1RAB9AMAOBROCK2MAP4K4
SCHEMBL15875686 0.81 MAOB (0.83) NPC1RAB9AMAOBROCK2MAP4K4
SCHEMBL15764676 0.81 NPC1 (1.00) NPC1RAB9AMAOBROCK2MAP4K4
SCHEMBL15764697 0.80 NPC1 (0.70) NPC1RAB9AMAOBROCK2MAP4K4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1708996-A1 FUSED HETEROYRAL DERIVATIVES FOR USE AS P38 KINASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2006-10-11 EP disclosed
WO-2005073189-A1 FUSED HETEROYRAL DERIVATIVES FOR USE AS P38 KINASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2005-08-11 WO disclosed