SCHEMBL5708155

SCHEMBL5708155

Cc1onc(-c2ccc(Cl)cc2)c1C(=O)Cl

nearest known ligand 0.66

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 11/20 0.66
GHSR Q92847 1/20 0.55
POLB P06746 1/20 0.54
NPC1 O15118 1/20 0.54
MEN1 O00255 2/20 0.53
KMT2A Q03164 2/20 0.53
MAPT P10636 1/20 0.53
GAA P10253 1/20 0.53
TSHR P16473 2/20 0.47
KDM4E B2RXH2 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11515850 0.89 GPBAR1 (0.59) GPBAR1POLBMEN1KMT2AGAA
SCHEMBL3548012 0.87 GPBAR1 (0.66) GPBAR1GHSRPOLBNPC1MEN1
SCHEMBL1575050 0.87 GPBAR1 (0.66) GPBAR1GHSRPOLBNPC1MEN1
SCHEMBL3068021 0.86 GPBAR1 (0.61) GPBAR1NPC1MEN1KMT2AGAA
SCHEMBL892042 0.85 KMT2A (0.71) GPBAR1POLBNPC1MEN1KMT2A
SCHEMBL11518716 0.83 GPBAR1 (0.48) GPBAR1MEN1KMT2AMAPTGAA
SCHEMBL11419174 0.83 GPBAR1 (0.61) GPBAR1GHSRPOLBNPC1MEN1
SCHEMBL3546359 0.83 GPBAR1 (0.78) GPBAR1GHSRPOLBNPC1
SCHEMBL2723582 0.83 GPBAR1 (0.62) GPBAR1POLBMEN1KMT2AMAPT
SCHEMBL11517320 0.82 GPBAR1 (0.66) GPBAR1GHSRPOLBNPC1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1706387-A1 SUBSTITUTED HETEROCYCLIC AMIDES HAVING A FUNGICIDAL EFFECT Bayer CropScience Aktiengesellschaft (DE) 2006-10-04 EP disclosed
WO-2005066138-A1 SUBSTITUTED HETEROCYCLIC AMIDES HAVING A FUNGICIDAL EFFECT BAYER CROPSCIENCE AG (DE) 2005-07-21 WO disclosed
US-4155905-A 6-Substituted penicillanic acid and derivatives thereof E. R. SQUIBB & SONS, INC. (US) 1979-05-22 US disclosed
US-4077967-A 6-Substituted penicillanic acid and derivatives thereof E. R. SQUIBB & SONS, INC. (US) 1978-03-07 US disclosed
US-4061851-A 7-Amino-7-arylthio cephalosporins E. R. SQUIBB & SONS, INC. (US) 1977-12-06 US disclosed
US-4061629-A 6-Amino-6-arylthio penicillanic acids and derivatives thereof E. R. SQUIBB & SONS, INC. (US) 1977-12-06 US disclosed
US-4029669-A 6-Benzalimino-6-arylthio penicillanic acids and derivatives thereof E. R. SQUIBB & SONS, INC. (US) 1977-06-14 US disclosed
US-4026886-A 7-Acyl-7-arylthiocephalosporins E. R. SQUIBB & SONS, INC. (US) 1977-05-31 US disclosed
US-3965093-A 6-Arylthio penicillanic acid and derivatives thereof E. R. SQUIBB & SONS, INC. (US) 1976-06-22 US disclosed
US-3954744-A ANTIBACTERIAL E. R. SQUIBB & SONS, INC. (US) 1976-05-04 US disclosed