SCHEMBL5712919

SCHEMBL5712919

CC(=O)N([C@H](C=O)CC(=O)O)N1C(=O)[C@@H](NC(=O)c2nccc3ccccc23)CC(=O)c2ccccc21

nearest known ligand 0.46

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 17/20 0.46
CASP8 Q14790 10/20 0.37
CASP3 P42574 2/20 0.35
DRD2 P14416 1/20 0.34
DRD3 P35462 1/20 0.34
RAB9A P51151 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL646096 0.87 CASP1 (0.46) CASP1CASP8CASP3DRD2DRD3
SCHEMBL5712985 0.86 CASP1 (0.48) CASP1
SCHEMBL646460 0.85 CASP1 (0.45) CASP1CASP8
SCHEMBL647010 0.83 CASP1 (0.43) CASP1CASP8DRD2DRD3
SCHEMBL7446425 0.80 CASP1 (0.32) CASP1
SCHEMBL648576 0.79 CASP1 (0.42) CASP1CASP8DRD2
SCHEMBL647046 0.79 CASP1 (0.43) CASP1CASP8CASP3
SCHEMBL644969 0.78 CASP1 (0.42) CASP1CASP8CASP3DRD2DRD3
SCHEMBL5712978 0.77 CASP1 (0.46) CASP1CASP8CASP3RAB9A
SCHEMBL8521265 0.77 CASP1 (0.46) CASP1CASP8CASP3RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0942925-B1 INHIBITORS OF INTERLEUKIN-1 BETA CONVERTING ENZYME VERTEX PHARMA (US) 2006-11-22 EP disclosed