SCHEMBL5712938

SCHEMBL5712938

CNCNc1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.52
ALDH1A1 P00352 4/20 0.52
MAPT P10636 3/20 0.52
L3MBTL1 Q9Y468 2/20 0.44
CYP3A4 P08684 3/20 0.44
KDM4E B2RXH2 1/20 0.44
TDP1 Q9NUW8 3/20 0.43
HSD17B10 Q99714 3/20 0.43
CTSD P07339 1/20 0.43
ATM Q13315 1/20 0.42
TAAR1 Q96RJ0 1/20 0.42
CYP1A2 P05177 2/20 0.42
CYP2C9 P11712 2/20 0.42
CYP2C19 P33261 2/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
HTT P42858 1/20 0.41
CA12 O43570 1/20 0.41
CA2 P00918 1/20 0.41
CA9 Q16790 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL16294582 0.97 MAPT (0.50) TSHRALDH1A1MAPTL3MBTL1CYP3A4
SCHEMBL43909 0.85 ALDH1A1 (0.60) TSHRALDH1A1MAPTL3MBTL1CYP3A4
SCHEMBL28937414 0.85 MAPT (0.41) TSHRALDH1A1MAPTL3MBTL1CYP3A4
Ammonia Solution, Strong SCHEMBL9517245 0.82 ALDH1A1 (0.57) TSHRALDH1A1MAPTL3MBTL1CYP3A4
SCHEMBL1759364 0.82 ALDH1A1 (0.57) TSHRALDH1A1MAPTL3MBTL1CYP3A4
Hydrochloric Acid SCHEMBL421277 0.80 ALDH1A1 (0.55) TSHRALDH1A1MAPTL3MBTL1CYP3A4
SCHEMBL1354067 0.79 MAPT (0.61) TSHRALDH1A1MAPTL3MBTL1CYP3A4
Sodium Chloride SCHEMBL421276 0.78 ALDH1A1 (0.52) TSHRALDH1A1MAPTL3MBTL1CYP3A4
Hydrochloric Acid SCHEMBL25404814 0.77 MAPT (0.58) TSHRALDH1A1MAPTL3MBTL1CYP3A4
SCHEMBL6017273 0.75 ALDH1A1 (0.77) TSHRALDH1A1MAPTL3MBTL1ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1727798-A1 NOVEL ARYL-CONTAINING 5-ACYLINDOLINONES, THE PRODUCTION THEREOF AND THEIR USE AS MEDICAMENTS Boehringer Ingelheim International GmbH (DE) 2006-12-06 EP disclosed
WO-2005087726-A1 NOVEL ARYL-CONTAINING 5-ACYLINDOLINONES, THE PRODUCTION THEREOF AND THEIR USE AS MEDICAMENTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2005-09-22 WO disclosed
EP-1115704-A1 NOVEL SUBSTITUTED INDOLINONES WITH AN INHIBITORY EFFECT ON VARIOUS KINASES AND CYCLIN/CDK COMPLEXES Boehringer Ingelheim Pharma KG (DE) 2001-07-18 EP disclosed
EP-0763524-B1 Urea and amide derivatives having ACAT inhibitory activity, their preparation and their therapeutic and prophylactic use SANKYO CO (JP) 2000-08-23 EP disclosed
WO-2000018734-A1 NOVEL SUBSTITUTED INDOLINONES WITH AN INHIBITORY EFFECT ON VARIOUS KINASES AND CYCLIN/CDK COMPLEXES BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-04-06 WO disclosed