SCHEMBL571364

SCHEMBL571364

O=S(=O)(O)c1ccc2nc[nH]c2c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKCI P41743 1/20 0.52
KDM4E B2RXH2 3/20 0.50
HDAC6 Q9UBN7 2/20 0.50
NAMPT P43490 2/20 0.50
MAPT P10636 2/20 0.50
CYP3A4 P08684 1/20 0.50
XDH P47989 1/20 0.50
RAD52 P43351 1/20 0.50
HTT P42858 2/20 0.49
SMN1; SMN2 Q16637 2/20 0.49
ALDH1A1 P00352 1/20 0.49
HPGD P15428 1/20 0.49
RAB9A P51151 1/20 0.49
MMP12 P39900 1/20 0.47
TDP1 Q9NUW8 2/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
CTNNB1 P35222 1/20 0.45
WNT3A P56704 1/20 0.45
FEN1 P39748 1/20 0.45
QPCT Q16769 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29724218 1.00 PRKCI (0.52) PRKCIKDM4EHDAC6NAMPTMAPT
Hydrochloric Acid SCHEMBL11090118 0.98 KDM4E (0.53) PRKCIKDM4EHDAC6NAMPTMAPT
Potassium SCHEMBL2918771 0.98 PRKCI (0.50) PRKCIKDM4EHDAC6NAMPTMAPT
Sulfurous Acid SCHEMBL9250718 0.91 PRKCI (0.44) PRKCIKDM4EHDAC6NAMPTMAPT
SCHEMBL571363 0.87 PRKCI (0.42) PRKCIKDM4EHDAC6NAMPTMAPT
SCHEMBL2918763 0.86 HDAC6 (0.41) PRKCIKDM4EHDAC6NAMPTMAPT
SCHEMBL28975737 0.86 HDAC6 (0.41) PRKCIKDM4EHDAC6NAMPTMAPT
SCHEMBL1266025 0.81 PRKCI (0.52) PRKCIKDM4EHDAC6NAMPTMAPT
SCHEMBL27786200 0.81 PRKCI (0.52) PRKCIKDM4EHDAC6NAMPTMAPT
SCHEMBL362001 0.81 POLB (0.58) PRKCIKDM4EHDAC6NAMPTMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 123 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021064116-A1 COMPOSITIONS WITH POLYMERIC OR OLIGOMERIC HYDROXY PHENYL TRIAZINE UV FILTER BASF SE (DE) 2021-04-08 WO claimed
CN-110540523-B Method for preparing sulfo-substituted benzimidazole and derivative thereof 安徽圣诺贝化学科技有限公司 2021-02-19 CN claimed
CN-110540523-A Method for preparing sulfo-substituted benzimidazole and derivative thereof ANHUI SHENGNUOBEI CHEMICAL TECH CO LTD 2019-12-06 CN claimed
CN-107955380-A LED display epoxy resin composition for packaging 李伟文 2018-04-24 CN claimed
EP-2941303-B1 NOVEL OIL-IN-WATER EMULSIONS RICH IN SALTS, HAVING HIGH VISCOSITY AND STABLE OVER TIME SOC D EXPL DE PRODUITS POUR LES IND CHIMIQUES SEPPIC (FR) 2017-05-10 EP claimed
EP-3105210-A1 BENZIMIDAZOL-2-AMINES AS MIDH1 INHIBITORS Bayer Pharma Aktiengesellschaft (DE) 2016-12-21 EP claimed
WO-2015121209-A1 BENZIMIDAZOL-2-AMINES AS MIDH1 INHIBITORS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2015-08-20 WO claimed
EP-0031473-B1 PROCESS FOR PREPARING 2-((ALKOXYCARBONYL)-AMINO)-5-(ALKYLTHIO)-1H-BENZIMIDAZOLES CHINOIN Gyogyszer és Vegyészeti Termékek Gyára RT. (HU) 1984-05-30 EP claimed
CN-118843451-A Cosmetic material 株式会社资生堂 2024-10-25 CN disclosed
WO-2024122465-A1 EMULSIFIED TOPICAL COMPOSITION AND METHOD FOR PRODUCING SAME ロート製薬株式会社 2024-06-13 WO disclosed
CN-117460490-A Skin external composition containing taurine crystal with useful component 考司美德制药株式会社 2024-01-26 CN disclosed
CN-117377454-A Skin care composition 考司美德制药株式会社 2024-01-09 CN disclosed
WO-2023210059-A1 DERMATOLOGICAL TOPICAL AGENT COMPOSITION CONTAINING USEFUL COMPONENT-INCLUDING TAURINE CRYSTALS コスメディ製薬株式会社 2023-11-02 WO disclosed
CN-113347959-B Cosmetic with white turbidity 株式会社资生堂 2023-10-27 CN disclosed
US-4659647-A BLEND WITH HYDROPHOBIC POLYMER AND STABILIZER MINNESOTA MINING AND MANUFACTURING COMPANY (US) 1987-04-21 US disclosed
EP-0185243-A2 Photosensitive silver halide material for obtaining half-tone black-and-white images and method for half-tone high-contrast reproduction MINNESOTA MINING AND MANUFACTURING COMPANY (US) 1986-06-25 EP disclosed
US-4517254-A ALKALI METAL HYDROXIDE, AMINOALKYLPOLYACID COMPOUNT SCHERING AKTIENGESELLSCHAFT (DE) 1985-05-14 US disclosed
EP-0139090-A1 Process for the pre-treatment of polyimides SCHERING AKTIENGESELLSCHAFT (DE) 1985-05-02 EP disclosed
US-4466805-A 1,1,6,6-TETRAALKOXY HEXA-2,4-DIENES MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1984-08-21 US disclosed
US-4248632-A ACTIVATION OF A POLYMER SURFACE WITH A PALLADIUM COMPLEX SALT SCHERING AKTIENGESELLSCHAFT (DE) 1981-02-03 US disclosed