SCHEMBL362001

SCHEMBL362001

NS(=O)(=O)c1ccc2nc[nH]c2c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.58
CASP6 P55212 1/20 0.58
CTDSP1 Q9GZU7 1/20 0.58
PRKCI P41743 1/20 0.56
KDM4E B2RXH2 3/20 0.55
MAPT P10636 2/20 0.55
RAD52 P43351 1/20 0.55
CYP3A4 P08684 1/20 0.50
NAMPT P43490 1/20 0.50
XDH P47989 1/20 0.50
CDK1 P06493 2/20 0.47
MMP12 P39900 1/20 0.47
CA1 P00915 2/20 0.47
CA2 P00918 2/20 0.47
CA12 O43570 1/20 0.47
CA3 P07451 1/20 0.47
CA4 P22748 1/20 0.47
CA6 P23280 1/20 0.47
CA5A P35218 1/20 0.47
CA7 P43166 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL362000 0.87 POLB (0.50) POLBCASP6CTDSP1PRKCIKDM4E
SCHEMBL4429286 0.81 PRKCI (0.52) POLBCASP6CTDSP1PRKCIKDM4E
SCHEMBL27786200 0.81 PRKCI (0.52) POLBCASP6CTDSP1PRKCIKDM4E
SCHEMBL571364 0.81 PRKCI (0.52) POLBCASP6CTDSP1PRKCIKDM4E
SCHEMBL29724218 0.81 PRKCI (0.52) POLBCASP6CTDSP1PRKCIKDM4E
SCHEMBL1266025 0.81 PRKCI (0.52) PRKCIKDM4EMAPTRAD52CYP3A4
Hydrochloric Acid SCHEMBL11090118 0.80 KDM4E (0.53) POLBCASP6CTDSP1PRKCIKDM4E
Potassium SCHEMBL2918771 0.80 PRKCI (0.50) POLBCASP6CTDSP1PRKCIKDM4E
SCHEMBL7174501 0.80 PARP1 (0.61) CA12CA9SMN1; SMN2
SCHEMBL11783649 0.79 MMP12 (0.49) PRKCIKDM4EMAPTRAD52CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 76 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105980365-B Benzimidazol-2-amines as mIDH1 inhibitors 拜耳医药股份公司 2019-06-21 CN claimed
EP-3407877-A1 NLRP3 INHIBITORS FOR THE TREATMENT OF INFLAMMATORY SKIN DISORDERS Galderma Research & Development (FR) 2018-12-05 EP claimed
EP-3233845-A1 PARG INHIBITORY COMPOUNDS Cancer Research Technology Limited (GB) 2017-10-25 EP claimed
CN-107295799-A Parg inhibiting compounds 癌症研究科技有限公司 2017-10-24 CN claimed
WO-2017129897-A1 NLRP3 INHIBITORS FOR THE TREATMENT OF INFLAMMATORY SKIN DISORDERS GALDERMA RESEARCH & DEVELOPMENT (FR) 2017-08-03 WO claimed
EP-3105210-A1 BENZIMIDAZOL-2-AMINES AS MIDH1 INHIBITORS Bayer Pharma Aktiengesellschaft (DE) 2016-12-21 EP claimed
WO-2016097749-A1 PARG INHIBITORY COMPOUNDS CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2016-06-23 WO claimed
WO-2015121209-A1 BENZIMIDAZOL-2-AMINES AS MIDH1 INHIBITORS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2015-08-20 WO claimed
EP-2744805-A1 HETEROARYL SODIUM CHANNEL INHIBITORS Amgen Inc. (US) 2014-06-25 EP claimed
WO-2013025883-A1 HETEROARYL SODIUM CHANNEL INHIBITORS AMGEN INC. (US) 2013-02-21 WO claimed
EP-2523559-A1 COMPOUNDS AND METHODS GlaxoSmithKline LLC (US) 2012-11-21 EP claimed
EP-2121656-A1 INHIBITORS OF SERINE PALMITOYLTRANSFERASE Pfizer Products Inc. (US) 2009-11-25 EP claimed
WO-2009007390-A2 2-PYRAZ INYLBENZ IMIDAZOLE DERIVATIVES AS RECEPTOR TYROSINE KINASE INHIBITORS ASTRAZENECA AB (SE) 2009-01-15 WO claimed
WO-2008084300-A1 INHIBITORS OF SERINE PALMITOYLTRANSFERASE PFIZER PRODUCTS INC. (US) 2008-07-17 WO claimed
EP-1879877-A2 ANTIMICROBIAL AGENTS Ranbaxy Laboratories Limited (IN) 2008-01-23 EP claimed
WO-2006117762-A2 ANTIMICROBIAL AGENTS RANBAXY LABORATORIES LIMITED (IN) 2006-11-09 WO claimed
US-12365681-B2 Dihydrobenzimidazolones for medical treatment C4 THERAPEUTICS, INC. (US) 2025-07-22 US disclosed
US-20250228824-A1 COMPOSITIONS AND METHODS FOR INHIBITION OF ITO AS TREATMENT FOR THE J WAVE SYNDROMES AND HYPOTHERMIA SIMON FRASER UNIVERSITY (CA) 2025-07-17 US disclosed
WO-2002032422-A2 EP4 RECEPTOR INHIBITORS TO TREAT RHEUMATOID ARTHRITIS PFIZER PHARMACEUTICALS INC. (JP) 2002-04-25 WO disclosed
WO-2002032900-A2 ARYL OR HETEROARYL FUSED IMIDAZOLE COMPOUNDS AS ANTI-INFLAMMATORY AND ANALGESIC AGENTS PFIZER PHARMACEUTICALS INC. (JP) 2002-04-25 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12365681-B2 Dihydrobenzimidazolones for medical treatment CRBN, CUL4A, ADRM1 POLB 2355/4885CASP6 3660/4885CTDSP1 2015/4885
US-20250228824-A1 COMPOSITIONS AND METHODS FOR INHIBITION OF ITO AS TREATMENT FOR THE J WAVE SYNDROMES AND HYPOTHERMIA KCNH2, KCNJ1, KCNJ8 POLB 3887/4885CASP6 2006/4885CTDSP1 3452/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.