Delprostenate

Delprostenate

SCHEMBL571387

COC(=O)/C=C/C/C=C\C[C@@H]1[C@@H](/C=C/[C@@H](O)COc2cccc(Cl)c2)[C@H](O)C[C@@H]1O

nearest known ligand 0.71

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Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PTGFR P43088 14/20 0.71
PTGER3 P43115 5/20 0.71
TBXA2R P21731 3/20 0.71
PTGER1 P34995 3/20 0.71
PTGER2 P43116 2/20 0.71
THRB P10828 1/20 0.71
ABCC4 O15439 2/20 0.69
ABCB11 O95342 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Delprostenate SCHEMBL8206607 0.92 ABCC4 (0.84) PTGFRPTGER3TBXA2RPTGER1PTGER2
SCHEMBL15389593 0.91 PTGFR (0.78) PTGFRPTGER3TBXA2RPTGER1PTGER2
SCHEMBL15389592 0.91 PTGFR (0.78) PTGFRPTGER3TBXA2RPTGER1PTGER2
SCHEMBL15389591 0.91 PTGFR (0.78) PTGFRPTGER3TBXA2RPTGER1PTGER2
Froxiprost SCHEMBL563113 0.88 PTGFR (0.72) PTGFRPTGER3TBXA2RPTGER1PTGER2
Cloprostenol SCHEMBL123596 0.83 PTGFR (1.00) PTGFRPTGER3TBXA2RPTGER1PTGER2
Cloprostenol SCHEMBL15669946 0.83 PTGFR (1.00) PTGFRPTGER3TBXA2RPTGER1PTGER2
Cloprostenol SCHEMBL14913508 0.83 PTGFR (1.00) PTGFRPTGER3TBXA2RPTGER1PTGER2
Cloprostenol SCHEMBL14913507 0.83 PTGFR (1.00) PTGFRPTGER3TBXA2RPTGER1PTGER2
Cloprostenol SCHEMBL17200671 0.83 PTGFR (1.00) PTGFRPTGER3TBXA2RPTGER1PTGER2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 131 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20160113942-A1 COMPOSITIONS COMPRISING A PROSTAGLANDIN FOR TREATING NEUROPSYCHIATRIC CONDITIONS INCEPTUM RESEARCH & THERAPEUTICS, INC. (CA) 2016-04-28 US claimed
US-9016221-B2 Surface topographies for non-toxic bioadhesion control UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2015-04-28 US claimed
EP-2667875-A1 COMPOSITIONS COMPRISING A PROSTAGLANDIN FOR TREATING NEUROPSYCHIATRIC CONDITIONS Inceptum Research & Therapeutics, Inc. (CA) 2013-12-04 EP claimed
US-20130309330-A1 COMPOSITIONS COMPRISING A PROSTAGLANDIN FOR TREATING NEUROPSYCHIATRIC CONDITIONS INCEPTUM RESEARCH & THERAPEUTICS, INC. (CA) 2013-11-21 US claimed
WO-2012100347-A1 COMPOSITIONS COMPRISING A PROSTAGLANDIN FOR TREATING NEUROPSYCHIATRIC CONDITIONS INCEPTUM RESEARCH & THERAPEUTICS, INC. (CA) 2012-08-02 WO claimed
US-20100226943-A1 SURFACE TOPOGRAPHIES FOR NON-TOXIC BIOADHESION CONTROL UNIVERSITY OF FLORIDA (US) 2010-09-09 US claimed
CN-101330905-A Freeze-drying process and products obtained thereby SCIDOSE LLC (US) 2008-12-24 CN claimed
EP-1954244-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY Scidose, Llc (US) 2008-08-13 EP claimed
WO-2007061529-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY SCIDOSE LLC. (US) 2007-05-31 WO claimed
US-20070116729-A1 Lyophilization process and products obtained thereby SCIDOSE LLC 2007-05-24 US claimed
WO-2000051617-A1 METHODS OF INCREASING BONE VOLUME USING NON-NATURALLY-OCCURRING FP SELECTIVE AGONISTS AND ANTIRESORPTIVE COMPOUNDS THE PROCTER & GAMBLE COMPANY (US) 2000-09-08 WO claimed
WO-2000051585-A2 USE OF A NON-NATURALLY-OCCURRING EP1 SELECTIVE AGONIST FOR INCREASING BONE VOLUME THE PROCTER & GAMBLE COMPANY (US) 2000-09-08 WO claimed
WO-1999012551-A1 METHOD OF INCREASING BONE VOLUME USING NON-NATURALLY-OCCURRING FP SELECTIVE AGONISTS THE PROCTER & GAMBLE COMPANY (US) 1999-03-18 WO claimed
WO-1999012550-A1 METHOD OF INCREASING BONE VOLUME THE PROCTER & GAMBLE COMPANY (US) 1999-03-18 WO claimed
EP-0664707-B1 COMBINATIONS OF PROSTAGLANDINS AND CLONIDINE DERIVATIVES FOR THE TREATMENT OF GLAUCOMA ALCON LAB INC (US) 1997-06-04 EP claimed
US-5605922-A VISION DISORDERS; SIDE EFFECT REDUCTION ALCON LABORATORIES, INC. (US) 1997-02-25 US claimed
WO-1996013267-A2 COMBINATIONS OF PROSTAGLANDINS AND BRIMONIDINE OR DERIVATIVES THEREOF FOR THE TREATMENT OF GLAUCOMA ALLERGAN (US) 1996-05-09 WO claimed
US-5480900-A Combinations of prostaglandins and clonidine derivatives for the treatment of glaucoma ALCON LABORATORIES, INC. (US) 1996-01-02 US claimed
EP-0664707-A1 COMBINATIONS OF PROSTAGLANDINS AND CLONIDINE DERIVATIVES FOR THE TREATMENT OF GLAUCOMA. ALCON LAB INC (US) 1995-08-02 EP claimed
WO-1994008585-A1 COMBINATIONS OF PROSTAGLANDINS AND CLONIDINE DERIVATIVES FOR THE TREATMENT OF GLAUCOMA ALCON LABORATORIES, INC. (US) 1994-04-28 WO claimed