SCHEMBL5717017

SCHEMBL5717017

CC[C@@]1(C(=O)O)CCCCN1S(=O)(=O)c1ccc(C(F)(F)F)cc1Cl

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 2/20 0.44
HCRTR2 O43614 2/20 0.44
ALDH1A1 P00352 2/20 0.44
MEN1 O00255 1/20 0.44
TSHR P16473 1/20 0.44
KMT2A Q03164 1/20 0.44
ATM Q13315 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
TRPV4 Q9HBA0 9/20 0.41
CCKBR P32239 1/20 0.40
SLC6A9 P48067 2/20 0.39
ERAP1 Q9NZ08 1/20 0.37
PPARD Q03181 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5717025 0.88 EPHX2 (0.44) HCRTR1HCRTR2ALDH1A1MEN1TSHR
SCHEMBL5716994 0.83 HCRTR1 (0.46) HCRTR1HCRTR2ALDH1A1MEN1TSHR
SCHEMBL5717206 0.83 ALDH1A1 (0.43) HCRTR1HCRTR2ALDH1A1TRPV4
SCHEMBL5717229 0.83 ALDH1A1 (0.43) HCRTR1HCRTR2ALDH1A1TRPV4
SCHEMBL11888834 0.73 MEN1 (0.50) HCRTR1HCRTR2ALDH1A1MEN1TSHR
SCHEMBL5717200 0.71 EPHX2 (0.46) HCRTR1HCRTR2ALDH1A1MEN1TSHR
SCHEMBL5717180 0.70 ITGB1 (0.38) ALDH1A1L3MBTL1
SCHEMBL5717014 0.70 ITGB1 (0.36) ALDH1A1MEN1KMT2A
SCHEMBL5717024 0.70 HCRTR1 (0.64) HCRTR1HCRTR2ALDH1A1MEN1TSHR
SCHEMBL5717057 0.69 HCRTR1 (0.60) HCRTR1HCRTR2ALDH1A1MEN1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1664010-A1 SULFONAMIDES ANTAGONISING N-TYPE CALCIUM CHANNELS Vernalis (R&D) Limited (GB) 2006-06-07 EP disclosed
WO-2005068448-A1 SULFONAMIDES ANTAGONISING N-TYPE CALCIUM CHANNELS IONIX PHARMACEUTICALS LIMITED (GB) 2005-07-28 WO disclosed