SCHEMBL5718320

SCHEMBL5718320

CC(c1ccc(-c2ccccc2)cc1)C1(O)CCC1

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.46
SLC6A2 P23975 1/20 0.42
SLC6A4 P31645 1/20 0.42
SLC6A3 Q01959 1/20 0.42
OPRM1 P35372 1/20 0.39
OPRD1 P41143 1/20 0.39
OPRK1 P41145 1/20 0.39
OPRL1 P41146 1/20 0.39
CYP17A1 P05093 1/20 0.38
ACP3 P15309 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5718317 0.95 SLC6A2 (0.49) PTGS2SLC6A2SLC6A4SLC6A3OPRM1
Hydrochloric Acid SCHEMBL5701112 0.93 SLC6A2 (0.47) PTGS2SLC6A2SLC6A4SLC6A3OPRM1
SCHEMBL19494132 0.89 OPRM1 (0.47) OPRM1OPRD1OPRK1OPRL1
SCHEMBL17086664 0.89 OPRM1 (0.47) OPRM1OPRD1OPRK1OPRL1
SCHEMBL17086651 0.89 OPRM1 (0.47) OPRM1OPRD1OPRK1OPRL1
SCHEMBL17086655 0.85 OPRM1 (0.47) SLC6A2SLC6A4OPRM1OPRD1OPRK1
SCHEMBL17086666 0.85 OPRM1 (0.47) SLC6A2SLC6A4OPRM1OPRD1OPRK1
SCHEMBL9717862 0.83 OPRM1 (0.46) SLC6A2SLC6A4SLC6A3OPRM1OPRD1
SCHEMBL8124662 0.83 OPRM1 (0.46) SLC6A2SLC6A4SLC6A3OPRM1OPRD1
SCHEMBL17086663 0.81 OPRM1 (0.50) OPRM1OPRD1OPRK1OPRL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1687288-A1 SUBSTITUTED ARYL CYCLOALKANOL DERIVATIVES AND METHODS OF THEIR USE Wyeth (US) 2006-08-09 EP claimed
WO-2005037809-A1 SUBSTITUTED ARYL CYCLOALKANOL DERIVATIVES AND METHODS OF THEIR USE WYETH (US) 2005-04-28 WO claimed
EP-1673059-A2 ALKANOL AND CYCLOALKANOL-AMINE DERIVATIVES AND METHODS OF THEIR USE Wyeth (US) 2006-06-28 EP disclosed
WO-2005037207-A2 ARYLALKYL-PIPERAZINE DERIVATIVES FOR THE TREATMENT OF CONDITIONS AMELIORATED BY MONOAMINE REUPTAKE INCLUDING VASOMOTOR SYMPTOMS (VMS) WYETH (US) 2005-04-28 WO disclosed