SCHEMBL5718429

SCHEMBL5718429

COc1cc(C#N)ccc1CONC(=O)c1ccccc1[AsH]Cc1ccnc(O)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
GPR6 P46095 2/20 0.35
HCRTR1 O43613 1/20 0.34
HCRTR2 O43614 1/20 0.34
NR3C2 P08235 1/20 0.34
SGMS2 Q8NHU3 1/20 0.34
L3MBTL1 Q9Y468 2/20 0.34
ATM Q13315 1/20 0.34
LRRK2 Q5S007 1/20 0.33
PDE5A O76074 1/20 0.33
PDE4A P27815 1/20 0.33
PDE4B Q07343 1/20 0.33
PDE4C Q08493 1/20 0.33
PDE4D Q08499 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
PDCD1 Q15116 1/20 0.32
CD274 Q9NZQ7 1/20 0.32
EGLN1 Q9GZT9 1/20 0.32
USP2 O75604 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1715722 0.85 TSHR (0.41) NPC1RAB9AGPR6LRRK2PDE5A
SCHEMBL12461145 0.77 PDE5A (0.41) PDE5APDCD1CD274USP2ALDH1A1
SCHEMBL1715615 0.76 POLB (0.44) NPC1RAB9AGPR6PDE5AALDH1A1
SCHEMBL1715115 0.75 KDR (0.47) PDE5A
SCHEMBL1715528 0.73 KIT (0.49) NR3C2PDE5ARXFP1GLATSHR
SCHEMBL12230044 0.72 TSHR (0.41) NPC1RAB9ANR3C2RXFP1ALDH1A1
SCHEMBL1714112 0.72 TSHR (0.41) NPC1RAB9APDE5APDE4APDE4B
SCHEMBL5718667 0.71 NR3C2 (0.40) NPC1RAB9AGPR6HCRTR1HCRTR2
SCHEMBL5718526 0.71 USP2 (0.35) NR3C2PDE5AUSP2ALDH1A1LMNA
SCHEMBL1715441 0.71 KDM4C (0.48) LRRK2PDE5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1697312-A2 HYDROXAMIC ACID ESTERS AND PHARMACEUTICAL USE THEREOF Leo Pharma A/S (DK) 2006-09-06 EP disclosed
WO-2005054179-A2 HYDROXAMIC ACID ESTERS AND PHARMACEUTICAL USE THEREOF LEO PHARMA A/S (DK) 2005-06-16 WO disclosed