SCHEMBL5718667

SCHEMBL5718667

CNC(=O)Nc1cc(Cc2c(N)cccc2C(=O)NOCc2ccc(C#N)cc2OC)ccn1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR3C2 P08235 5/20 0.40
KIT P10721 1/20 0.34
BRAF P15056 1/20 0.34
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34
SGMS2 Q8NHU3 1/20 0.33
GPR6 P46095 1/20 0.33
HCRTR1 O43613 1/20 0.33
HCRTR2 O43614 1/20 0.33
USP2 O75604 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
TP53 P04637 1/20 0.33
CYP1A2 P05177 1/20 0.33
GLA P06280 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
TSHR P16473 1/20 0.33
CYP2C19 P33261 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1715528 0.85 KIT (0.49) NR3C2KITBRAFGLATSHR
SCHEMBL12461798 0.75 KIT (0.51) NR3C2KITBRAFNPC1RAB9A
SCHEMBL1716023 0.72 KIT (0.53) KITBRAFGLAGCKMEN1
SCHEMBL1715722 0.71 TSHR (0.41) KITBRAFNPC1RAB9AGPR6
SCHEMBL5718429 0.71 NPC1 (0.37) NR3C2NPC1RAB9ASGMS2GPR6
SCHEMBL1715115 0.71 KDR (0.47) KITBRAF
SCHEMBL1715615 0.71 POLB (0.44) KITBRAFNPC1RAB9AGPR6
SCHEMBL1715441 0.67 KDM4C (0.48)
SCHEMBL1714112 0.67 TSHR (0.41) NPC1RAB9ATSHR
SCHEMBL1490730 0.66 GCK (0.54) BRAFNPC1RAB9ATP53GCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1697312-A2 HYDROXAMIC ACID ESTERS AND PHARMACEUTICAL USE THEREOF Leo Pharma A/S (DK) 2006-09-06 EP disclosed
WO-2005054179-A2 HYDROXAMIC ACID ESTERS AND PHARMACEUTICAL USE THEREOF LEO PHARMA A/S (DK) 2005-06-16 WO disclosed