SCHEMBL572074

SCHEMBL572074

CCC(C)C(NC(=O)OC(C)(C)C)C(=O)NC(CC(=O)O)Cc1ccc(F)c(F)c1F

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSS P25774 2/20 0.47
CTSK P43235 2/20 0.47
CA2 P00918 2/20 0.42
PSENEN Q9NZ42 1/20 0.41
CTSD P07339 3/20 0.40
HDAC3 O15379 1/20 0.39
HDAC4 P56524 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC7 Q8WUI4 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC10 Q969S8 1/20 0.39
HDAC11 Q96DB2 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
HDAC9 Q9UKV0 1/20 0.39
HDAC5 Q9UQL6 1/20 0.39
KDM4E B2RXH2 3/20 0.39
HTT P42858 1/20 0.39
ALDH1A1 P00352 2/20 0.38
HPGD P15428 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3995181 0.87 ATM (0.44) CTSSCTSK
SCHEMBL14982900 0.86 CTSS (0.48) CTSSCTSKCA2PSENENCTSD
SCHEMBL572076 0.86 CTSS (0.48) CTSSCTSKCA2PSENENCTSD
SCHEMBL572951 0.81 CTSS (0.53) CTSSCTSK
SCHEMBL10057465 0.78 CTSS (0.45) CTSSCTSKCA2PSENENCTSD
SCHEMBL572131 0.78 CTSS (0.45) CTSSCTSKCA2PSENENCTSD
SCHEMBL4893696 0.77 CTSS (0.50) CTSSCTSK
SCHEMBL13905757 0.76 ATM (0.43) CTSSCTSKHDAC3HDAC4HDAC1
SCHEMBL12394647 0.74 CTSS (0.44) CTSSCTSK
SCHEMBL7094300 0.73 CTSS (0.53) CTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2600888-A2 NOVEL COMPOUNDS AS DPP-IV INHIBITORS AND PROCESS FOR PREPARATION THEREOF Cadila Pharmaceuticals Ltd. (IN) 2013-06-12 EP disclosed
WO-2012017391-A2 NOVEL COMPOUNDS AS DPP-IV INHIBITORS AND PROCESS FOR PREPARATION THEREOF CADILA PHARMACEUTICALS LIMITED (IN) 2012-02-09 WO disclosed