SCHEMBL5723243

SCHEMBL5723243

O=C(NNC(=O)[C@@H]1C[C@@H](S)CN1S(=O)(=O)c1ccc2ccccc2c1)Nc1ccccc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ECE1 P42892 7/20 0.59
MME P08473 2/20 0.59
ACE P12821 2/20 0.59
HCRTR1 O43613 1/20 0.48
HCRTR2 O43614 1/20 0.48
EIF2AK3 Q9NZJ5 1/20 0.47
MAPT P10636 2/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
CA2 P00918 1/20 0.42
AKR1C3 P42330 4/20 0.42
AKR1C1 Q04828 1/20 0.41
CCR4 P51679 2/20 0.41
BRD4 O60885 1/20 0.39
LMNA P02545 2/20 0.39
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 1/20 0.39
ALDH1A1 P00352 1/20 0.39
TP53 P04637 1/20 0.39
ALOX15 P16050 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5723245 1.00 ECE1 (0.59) ECE1MMEACEHCRTR1HCRTR2
SCHEMBL5724183 0.91 ECE1 (0.54) ECE1MMEACEHCRTR1HCRTR2
SCHEMBL5723246 0.90 ECE1 (0.63) ECE1MMEACEHCRTR1HCRTR2
Dimethylamine SCHEMBL5724587 0.86 ECE1 (0.66) ECE1MMEACEHCRTR1HCRTR2
SCHEMBL5723488 0.86 ECE1 (0.66) ECE1MMEACEHCRTR1HCRTR2
SCHEMBL5723097 0.85 ECE1 (0.67) ECE1MMEACEHCRTR1HCRTR2
SCHEMBL7142911 0.84 ECE1 (0.61) ECE1MMEACEHCRTR1HCRTR2
SCHEMBL7142916 0.84 ECE1 (0.61) ECE1MMEACEHCRTR1HCRTR2
SCHEMBL5722964 0.84 ECE1 (0.64) ECE1MMEACEHCRTR1HCRTR2
SCHEMBL5722970 0.84 ECE1 (0.64) ECE1MMEACEHCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1317428-B1 PYRROLIDINE-2-CARBOXYLIC ACID HYDRAZIDE DERIVATIVES FOR USE AS METALLOPROTEASE INHIBITORS HOFFMANN LA ROCHE (CH) 2006-04-19 EP disclosed