SCHEMBL5723488

SCHEMBL5723488

CC(=O)NNC(=O)[C@@H]1C[C@@H](S)CN1S(=O)(=O)c1ccc2ccccc2c1

nearest known ligand 0.66

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ECE1 P42892 10/20 0.66
MME P08473 2/20 0.66
ACE P12821 2/20 0.66
EIF2AK3 Q9NZJ5 1/20 0.50
HCRTR1 O43613 1/20 0.47
HCRTR2 O43614 1/20 0.47
LMNA P02545 2/20 0.43
ALDH1A1 P00352 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
CCR4 P51679 3/20 0.43
AKR1C3 P42330 3/20 0.43
AKR1C1 Q04828 1/20 0.42
HPGD P15428 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5723097 0.90 ECE1 (0.67) ECE1MMEACEEIF2AK3HCRTR1
SCHEMBL5722964 0.90 ECE1 (0.64) ECE1MMEACEEIF2AK3HCRTR1
Dimethylamine SCHEMBL5724587 0.90 ECE1 (0.66) ECE1MMEACEEIF2AK3HCRTR1
SCHEMBL5722970 0.90 ECE1 (0.64) ECE1MMEACEEIF2AK3HCRTR1
SCHEMBL5723246 0.87 ECE1 (0.63) ECE1MMEACEEIF2AK3HCRTR1
SCHEMBL7148134 0.87 ECE1 (0.64) ECE1MMEACEEIF2AK3HCRTR1
SCHEMBL7148136 0.87 ECE1 (0.64) ECE1MMEACEEIF2AK3HCRTR1
SCHEMBL5723745 0.86 ECE1 (0.70) ECE1MMEACEEIF2AK3HCRTR1
SCHEMBL5723245 0.86 ECE1 (0.59) ECE1MMEACEEIF2AK3HCRTR1
SCHEMBL5723243 0.86 ECE1 (0.59) ECE1MMEACEEIF2AK3HCRTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1317428-B1 PYRROLIDINE-2-CARBOXYLIC ACID HYDRAZIDE DERIVATIVES FOR USE AS METALLOPROTEASE INHIBITORS HOFFMANN LA ROCHE (CH) 2006-04-19 EP disclosed