SCHEMBL5723317

SCHEMBL5723317

C#CCOc1nc(Nc2ccc(S(N)(=O)=O)cc2)ncc1C#N

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 11/20 0.59
CDK1 P06493 7/20 0.59
CCNB1 P14635 2/20 0.59
KDR P35968 3/20 0.56
CA2 P00918 4/20 0.53
CCNA2 P20248 5/20 0.52
CCNA1 P78396 5/20 0.52
CCNT1 O60563 2/20 0.52
CDK9 P50750 2/20 0.52
IKBKB O14920 2/20 0.47
CA1 P00915 3/20 0.46
CA9 Q16790 3/20 0.46
CA4 P22748 2/20 0.46
CA12 O43570 1/20 0.46
CA7 P43166 1/20 0.46
CDK7 P50613 1/20 0.45
CCNH P51946 1/20 0.45
CDC7 O00311 1/20 0.43
PLK4 O00444 1/20 0.43
CHEK1 O14757 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5723276 0.88 CDK1 (0.57) CDK2CDK1CCNB1KDRCA2
SCHEMBL5723409 0.87 CDK1 (0.56) CDK2CDK1CCNB1KDRCA2
SCHEMBL25665758 0.87 CDK2 (0.60) CDK2CDK1CCNB1KDRCA2
SCHEMBL5723191 0.86 CDK2 (0.55) CDK2CDK1CCNB1KDRCA2
SCHEMBL1474324 0.85 CDK2 (0.56) CDK2CDK1CCNB1KDRCA2
SCHEMBL24477952 0.84 CDK2 (0.59) CDK2CDK1CCNB1KDRCA2
SCHEMBL5723725 0.84 CDK2 (0.50) CDK2CDK1CCNB1KDRCA2
SCHEMBL5723688 0.83 CDK2 (0.56) CDK2CDK1CCNB1KDRCA2
SCHEMBL5723476 0.83 CDK2 (0.49) CDK2CDK1CCNB1KDRCA2
SCHEMBL5723568 0.82 CDK2 (0.51) CDK2CDK1CCNB1KDRCCNA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1406876-B1 2-ANILINO-PYRIMIDINE DERIVATIVES AS CYCLIN DEPENDENT KINASE INHIBITORS ASTRAZENECA AB (SE) 2006-12-27 EP disclosed