SCHEMBL5723409

SCHEMBL5723409

C#CCOc1nc(Nc2ccc(S(=O)(=O)NC)cc2)ncc1C#N

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 12/20 0.56
CDK2 P24941 11/20 0.56
KDR P35968 7/20 0.56
CCNA2 P20248 6/20 0.46
CCNT1 O60563 5/20 0.46
CDK9 P50750 5/20 0.46
CCNA1 P78396 5/20 0.46
CCNB1 P14635 4/20 0.46
CDK7 P50613 2/20 0.43
CCNH P51946 2/20 0.43
CDK5 Q00535 1/20 0.43
CDK5R1 Q15078 1/20 0.43
CA2 P00918 1/20 0.42
CCNB2 O95067 1/20 0.42
CCNB3 Q8WWL7 1/20 0.42
PTK2 Q05397 1/20 0.40
AURKA O14965 1/20 0.40
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
PLK1 P53350 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5723276 0.88 CDK1 (0.57) CDK1CDK2KDRCCNA2CCNT1
SCHEMBL5723317 0.87 CDK2 (0.59) CDK1CDK2KDRCCNA2CCNT1
SCHEMBL5723191 0.87 CDK2 (0.55) CDK1CDK2KDRCCNA2CCNT1
SCHEMBL5723568 0.86 CDK2 (0.51) CDK1CDK2KDRCCNA2CCNT1
SCHEMBL5723725 0.86 CDK2 (0.50) CDK1CDK2KDRCCNA2CCNT1
SCHEMBL24477749 0.86 CDK2 (0.50) CDK1CDK2KDRCCNA2CCNT1
SCHEMBL5723688 0.85 CDK2 (0.56) CDK1CDK2KDRCCNA2CCNT1
SCHEMBL5723476 0.85 CDK2 (0.49) CDK1CDK2KDRCCNA2CCNT1
SCHEMBL5723609 0.85 CDK2 (0.49) CDK1CDK2KDRCCNA2CCNT1
SCHEMBL5723722 0.84 CDK2 (0.48) CDK1CDK2KDRCCNA2CCNT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1406876-B1 2-ANILINO-PYRIMIDINE DERIVATIVES AS CYCLIN DEPENDENT KINASE INHIBITORS ASTRAZENECA AB (SE) 2006-12-27 EP disclosed