SCHEMBL5723391

SCHEMBL5723391

COc1cccc(C(=O)c2cc3c(cc2-c2ccc(S(C)(=O)=O)cc2)OCO3)c1

nearest known ligand 0.74

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 8/20 0.74
PTGS1 P23219 2/20 0.74
CYP2C8 P10632 1/20 0.50
CTNNB1 P35222 1/20 0.49
WNT3A P56704 1/20 0.49
MAPT P10636 2/20 0.44
EDNRB P24530 1/20 0.44
EDNRA P25101 1/20 0.44
STS P08842 1/20 0.44
KDM4E B2RXH2 2/20 0.43
LMNA P02545 2/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
POLB P06746 1/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
TP53 P04637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5723370 0.86 PTGS2 (0.78) PTGS2PTGS1MAPTLMNAKMT2A
SCHEMBL5723316 0.85 PTGS2 (0.77) PTGS2PTGS1
SCHEMBL5723358 0.85 PTGS2 (1.00) PTGS2PTGS1CTNNB1WNT3ATP53
SCHEMBL6732299 0.83 PTGS2 (0.62) PTGS2PTGS1MAPTNPC1RAB9A
SCHEMBL5724506 0.80 PTGS2 (0.69) PTGS2PTGS1NPC1RAB9A
SCHEMBL5723269 0.80 PTGS2 (0.73) PTGS2PTGS1EDNRBEDNRAKDM4E
SCHEMBL6730868 0.79 PTGS2 (0.70) PTGS2PTGS1MAPTEDNRBEDNRA
SCHEMBL5723481 0.79 PTGS2 (0.81) PTGS2PTGS1
SCHEMBL5723355 0.78 PTGS2 (0.48) PTGS2PTGS1MAPTKDM4EMEN1
SCHEMBL5723040 0.77 PTGS2 (0.49) PTGS2PTGS1CTNNB1WNT3AEDNRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1406609-B1 SUBSTITUTED ARYL COMPOUNDS AS NOVEL CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE NITROMED INC (US) 2006-09-06 EP claimed
US-6706724-B2 ANTITUMOR AGENTS; ANTIINFLAMMATORY AGENTS; ANALGESICS; ANTIPYRETIC AGENT NITROMED, INC. 2004-03-16 US claimed
US-6706724-B2 ANTITUMOR AGENTS; ANTIINFLAMMATORY AGENTS; ANALGESICS; ANTIPYRETIC AGENT NITROMED, INC. 2004-03-16 US disclosed